日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Functional analysis of JPH2-knockout cardiomyocytes identifies ECCD as a novel indicator in a human cardiac modelJPH2

对 JPH2 敲除心肌细胞的功能分析表明,ECCD 是人类心脏模型中的一种新型指标。

Tianwei Guo #,Hongyue Wang #,Fujian Wu #,Wenjing Lu,Min Zhu,Shuhong Ma,Yongshuai Zhang,Yuting Yan,Meng Zhou,Didaer Talanaite,Siyu Liu,Man Qi,Feng Lan,Xujie Liu

Treatment with L-type amino acid transporter 1 inhibitor JPH203 enhances protein synthesis in C2C12 myotubes.

用 L 型氨基酸转运体 1 抑制剂 JPH203 治疗可增强 C2C12 肌管中的蛋白质合成。

Takegaki Junya, Saneyasu Takaoki, Honda Kazuhisa

Functional characterization of a novel JPH2 variant (p.R160H) associated with dilated cardiomyopathy

对一种与扩张型心肌病相关的新型JPH2变异体(p.R160H)进行功能表征

Jiao, Kailu; Gong, Ke; Luo, Yong; Liu, RuiLin; Wang, Lei; Yao, Yao; Xie, Li

Structural basis for the inhibition mechanism of LAT1-4F2hc complex by JPH203

JPH203抑制LAT1-4F2hc复合物的结构基础

Hu, Ziwei; Yan, Renhong

L-type amino acid transporter 1 inhibitor JPH203 prevents the growth of cabazitaxel-resistant prostate cancer by inhibiting cyclin-dependent kinase activity

L型氨基酸转运蛋白1抑制剂JPH203通过抑制细胞周期蛋白依赖性激酶活性来阻止卡巴他赛耐药性前列腺癌的生长。

Rii, Junryo; Sakamoto, Shinichi; Mizokami, Atsushi; Xu, Minhui; Fujimoto, Ayumi; Saito, Shinpei; Koike, Hidekazu; Tamura, Takaaki; Arai, Takayuki; Yamada, Yasutaka; Goto, Yusuke; Sazuka, Tomokazu; Imamura, Yusuke; Suzuki, Kazuhiro; Kanai, Yoshikatsu; Anzai, Naohiko; Ichikawa, Tomohiko

The LAT1 inhibitor JPH203 suppresses the growth of castration-resistant prostate cancer through a CD24-mediated mechanism

LAT1抑制剂JPH203通过CD24介导的机制抑制去势抵抗性前列腺癌的生长。

Saito, Shinpei; Ando, Keisuke; Sakamoto, Shinichi; Xu, Minhui; Yamada, Yasutaka; Rii, Junryo; Kanaoka, Sanji; Wei, Jiaxing; Zhao, Xue; Pae, Sangjon; Kanesaka, Manato; Goto, Yusuke; Sazuka, Tomokazu; Imamura, Yusuke; Reien, Yoshie; Hamaguchi-Suzuki, Norie; Saito, Shota; Hirayama, Yuri; Hashimoto, Hirofumi; Kanai, Yoshikatsu; Ichikawa, Tomohiko; Anzai, Naohiko

Insights into the Transport Cycle of LAT1 and Interaction with the Inhibitor JPH203

LAT1转运周期及其与抑制剂JPH203相互作用的研究进展

Brunocilla, Chiara; Console, Lara; Rovella, Filomena; Indiveri, Cesare

The Junctophilin-2 Mutation p.(Thr161Lys) Is Associated with Hypertrophic Cardiomyopathy Using Patient-Specific iPS Cardiomyocytes and Demonstrates Prolonged Action Potential and Increased Arrhythmogenicity

Junctophilin-2 突变 p.(Thr161Lys) 与使用患者特异性 iPS 心肌细胞的肥厚性心肌病有关,并表现出动作电位延长和心律失常性增加

Joona Valtonen, Chandra Prajapati, Reeja Maria Cherian, Sari Vanninen, Marisa Ojala, Krista Leivo, Tiina Heliö, Juha Koskenvuo, Katriina Aalto-Setälä

LAT1 inhibitor JPH203 sensitizes cancer cells to radiation by enhancing radiation-induced cellular senescence

LAT1抑制剂JPH203通过增强辐射诱导的细胞衰老来提高癌细胞对辐射的敏感性。

Bo, Tomoki; Kobayashi, Sho; Inanami, Osamu; Fujii, Junichi; Nakajima, Osamu; Ito, Tsunekata; Yasui, Hironobu

Pachymic Acid Attenuated Doxorubicin-Induced Heart Failure by Suppressing miR-24 and Preserving Cardiac Junctophilin-2 in Rats

茯苓酸通过抑制 miR-24 和保护大鼠心脏连接蛋白-2 减轻阿霉素诱发的心力衰竭

Nahla N Younis, Alaa Salama, Mohamed A Shaheen, Rana G Eissa