日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Association Between Genetic Polymorphisms of UGT1A1, ABCG2, and NR1I2 and Dolutegravir Pharmacokinetic Parameters in Thai People Living with HIV

UGT1A1、ABCG2 和 NR1I2 基因多态性与泰国 HIV 感染者多替拉韦药代动力学参数的关联性研究

Chanruang, Anan; Birnbaum, Angela K; Sirilun, Sasithorn; Chupradit, Suthunya; Ubolyam, Sasiwimol; Hiranburana, Napon; Cho, Yong Soon; Shin, Jae Gook; Avihingsanon, Anchalee; Punyawudho, Baralee

Association of NR1I2 Polymorphism with Midazolam Clearance in Mechanically Ventilated ICU Patients: A Population Pharmacokinetic and Pharmacogenetic Study

NR1I2多态性与机械通气ICU患者咪达唑仑清除率的相关性:一项群体药代动力学和药物遗传学研究

Xie, Helin; Zheng, You; Zhang, Hui; Guo, Yanmei; Liu, Maobai; Weng, Qinyong; Wu, Xuemei

A bromodomain-independent mechanism of gene regulation by the BET inhibitor JQ1: direct activation of nuclear receptor PXR

BET 抑制剂 JQ1 的不依赖溴结构域的基因调控机制:直接激活核受体 PXR

Andrew D Huber, Shyaron Poudel, Jing Wu, Darcie J Miller, Wenwei Lin, Lei Yang, Monicah N Bwayi, Mary Ashley Rimmer, Rebecca R Florke Gee, Jayaraman Seetharaman, Sergio C Chai, Taosheng Chen

NR1I2 as a core biological target in chronic venous ulcer tissues treated with ultrasound therapy

NR1I2是超声治疗慢性静脉溃疡组织的核心生物靶点

Lu, Chuanyingzi; Zhang, Jingli; Zhang, Yajing; Bao, Xiaoshi

The F-box-only protein 44 regulates pregnane X receptor protein level by ubiquitination and degradation

F-box 独有蛋白 44 通过泛素化和降解调节孕烷 X 受体蛋白水平

Rebecca R Florke Gee, Andrew D Huber, Jing Wu, Richa Bajpai, Allister J Loughran, Shondra M Pruett-Miller, Taosheng Chen

Molecular basis of crosstalk in nuclear receptors: heterodimerization between PXR and CAR and the implication in gene regulation

核受体串扰的分子基础:PXR 和 CAR 之间的异二聚化及其对基因调控的影响

Monicah N Bwayi, Efren Garcia-Maldonado, Sergio C Chai, Boer Xie, Shirish Chodankar, Andrew D Huber, Jing Wu, Kavya Annu, William C Wright, Hyeong-Min Lee, Jayaraman Seetharaman, Jingheng Wang, Cameron D Buchman, Junmin Peng, Taosheng Chen

Combination of Paclitaxel and PXR Antagonist SPA70 Reverses Paclitaxel-Resistant Non-Small Cell Lung Cancer

紫杉醇与 PXR 拮抗剂 SPA70 联合治疗可逆转紫杉醇耐药性非小细胞肺癌

Xiaxia Niu, Ting Wu, Qishuang Yin, Xinsheng Gu, Gege Li, Changlong Zhou, Mei Ma, Li Su, Shu Tang, Yanan Tian, Ming Yang, Hongmei Cui

Effects of NR1I2 and ABCB1 Genetic Polymorphisms on Everolimus Pharmacokinetics in Japanese Renal Transplant Patients

NR1I2 和 ABCB1 基因多态性对日本肾移植患者依维莫司药代动力学的影响

Yagishita, Hironobu; Kagaya, Hideaki; Saito, Mitsuru; Numakura, Kazuyuki; Yamamoto, Ryohei; Sagehashi, Ryuichiro; Habuchi, Tomonori; Satoh, Shigeru; Miura, Masatomo

Nuclear Receptor PXR Confers Irradiation Resistance by Promoting DNA Damage Response Through Stabilization of ATF3

核受体 PXR 通过稳定 ATF3 促进 DNA 损伤反应,从而赋予抗辐射能力

Xiaxia Niu, Hongmei Cui, Xinsheng Gu, Ting Wu, Min Sun, Changlong Zhou, Mei Ma

Mice blocking Ser347 phosphorylation of pregnane x receptor develop hepatic fasting-induced steatosis and hypertriglyceridemia

阻断孕烷 x 受体 Ser347 磷酸化的小鼠发生肝脏禁食诱发脂肪变性和高甘油三酯血症

Kosuke Yokobori, Artiom Gruzdev, Masahiko Negishi