日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Role of PDE3A in Cancer

PDE3A在癌症中的作用

Pu, Shengyu; Zhang, Qihe; Miao, Mi; Chen, Bohong; Xu, Jiarui; Lei, Jingyi; Tang, Xiaojiang; Hao, Na

Pan-cancer ex vivo target evaluation of phosphodiesterase 3 A (PDE3A)

磷酸二酯酶 3A (PDE3A) 的泛癌体外靶点评价

Rice, Kiesha; Lehtinen, Noora; Välimäki, Eetu; Suhonen, Janne; Taimen, Pekka; Kettunen, Kimmo; Ventelä, Sami; Kononen, Juha; Sihto, Harri; Rantala, Juha K

PDE3A as a Therapeutic Target for the Modulation of Compartmentalised Cyclic Nucleotide-Dependent Signalling

PDE3A作为调节区室化环核苷酸依赖性信号传导的治疗靶点

Pati, Swaroop Ranjan; Sholokh, Anastasiia; Klussmann, Enno

First-in-Human Dose-Escalation Study of the First-in-Class PDE3A-SLFN12 Complex Inducer BAY 2666605 in Patients with Advanced Solid Tumors Coexpressing SLFN12 and PDE3A

首个PDE3A-SLFN12复合物诱导剂BAY 2666605在共表达SLFN12和PDE3A的晚期实体瘤患者中的首次人体剂量递增研究

Kyriakos P Papadopoulos ,Meredith McKean ,Silvia Goldoni ,Isabelle Genvresse ,Marine F Garrido ,Rui Li ,Gary Wilkinson ,Christoph Kneip ,Timothy A Yap

Discovery of BAY 2666605, a Molecular Glue for PDE3A and SLFN12

BAY 2666605 的发现,一种 PDE3A 和 SLFN12 的分子胶

Lewis, Timothy A; Ellermann, Manuel; Kopitz, Charlotte; Lange, Martin; de Waal, Luc; Wu, Xiaoyun; Tersteegen, Adrian; Denner, Karsten; Lienau, Philip; Kaulfuss, Stefan; Goldoni, Silvia; Meyerson, Matthew; Greulich, Heidi; Gradl, Stefan N

Velcrin molecular glues induce apoptosis in glioblastomas with high PDE3A and SLFN12 expression

Velcrin 分子胶可诱导 PDE3A 和 SLFN12 表达较高的胶质母细胞瘤细胞凋亡

Elisa Aquilanti, Silvia Goldoni, Andrew Baker, Kristyna Kotynkova, Sawyer Andersen, Vincent Bozinov, Galen F Gao, Andrew D Cherniack, Martin Lange, Ralf Lesche, Charlotte Kopitz, Philip Lienau, Timothy A Lewis, Marine Garrido, Stefan Gradl, Henrik Seidel, Yuen-Yi Tseng, Keith L Ligon, Patrick Y Wen,

Integrated Proteomics Unveils Nuclear PDE3A2 as a Regulator of Cardiac Myocyte Hypertrophy

综合蛋白质组学揭示核 PDE3A2 作为心肌细胞肥大的调节剂

Gunasekaran Subramaniam #, Katharina Schleicher #, Duangnapa Kovanich #, Anna Zerio, Milda Folkmanaite, Ying-Chi Chao, Nicoletta C Surdo, Andreas Koschinski, Jianshu Hu, Arjen Scholten, Albert J R Heck, Maria Ercu, Anastasiia Sholokh, Kyung Chan Park, Enno Klussmann, Viviana Meraviglia, Milena Belli

PDE3A and GSK3B as Atrial Fibrillation Susceptibility Genes in the Chinese Population via Bioinformatics and Genome-Wide Association Analysis

通过生物信息学和全基因组关联分析,探讨PDE3A和GSK3B作为中国人群房颤易感基因的作用

Zhou, Zechen; Wang, Yu; Li, Xiaoyi; Zhang, Yinan; Yuan, Lichuang; Chen, Dafang; Wang, Xuedong

Structure of PDE3A-SLFN12 complex reveals requirements for activation of SLFN12 RNase

PDE3A-SLFN12复合物的结构揭示了SLFN12 RNase激活的必要条件

Colin W Garvie #,Xiaoyun Wu #,Malvina Papanastasiou,Sooncheol Lee,James Fuller,Gavin R Schnitzler,Steven W Horner,Andrew Baker,Terry Zhang,James P Mullahoo,Lindsay Westlake,Stephanie H Hoyt,Marcus Toetzl,Matthew J Ranaghan,Luc de Waal,Joseph McGaunn,Bethany Kaplan,Federica Piccioni,Xiaoping Yang,Martin Lange,Adrian Tersteegen,Donald Raymond,Timothy A Lewis,Steven A Carr,Andrew D Cherniack,Christopher T Lemke,Matthew Meyerson,Heidi Greulich

Structure of PDE3A-SLFN12 complex and structure-based design for a potent apoptosis inducer of tumor cells

PDE3A-SLFN12 复合物的结构和基于结构的设计用于有效的肿瘤细胞凋亡诱导剂

Jie Chen #, Nan Liu #, Yinpin Huang #, Yuanxun Wang #, Yuxing Sun #, Qingcui Wu, Dianrong Li, Shuanhu Gao, Hong-Wei Wang, Niu Huang, Xiangbing Qi, Xiaodong Wang