日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Genetic variations in AAK1 and ADAM17 associated with circulatory cytokines changes influence COVID-19 susceptibility and severity

与循环细胞因子变化相关的AAK1和ADAM17基因变异会影响COVID-19的易感性和严重程度。

Bouzid, Amal; Elemam, Noha M; Alsafar, Habiba; Venkatachalam, Thenmozhi; Eldoahji, Leen; Halabi, Nour; Saleh, Mohamed A; Talaat, Iman M; Taneera, Jalal; Sulaiman, Nabil; Maghazachi, Azzam A; Hamid, Qutayba; Hamoudi, Rifat; Saber-Ayad, Maha

AAK1 activation-mediated iron trafficking drives ferroptotic cell death.

AAK1 激活介导的铁转运驱动铁死亡。

Development of pyrazolo[1,5-a]pyrimidine based macrocyclic kinase inhibitors targeting AAK1.

开发以吡唑并[1,5-a]嘧啶为基础的大环激酶抑制剂,靶向AAK1。

Mensing Theresa E, Kurz Christian G, Amrhein Jennifer A, Ehret Theresa A L, Preuss Franziska, Mathea Sebastian, Karim Marwah, Tran Do Hoang Nhu, Kadlecova Zuzana, Tolvanen Tuomas A, Martinez-Molina Daniel, Müller Susanne, Einav Shirit, Knapp Stefan, Hanke Thomas

Synthesis, Experimental and Computational Evaluation of SERAAK1 as a 5-HT(2A) Receptor Ligand

SERAAK1作为5-HT(2A)受体配体的合成、实验和计算评价

Zięba, Agata; Kędzierska, Ewa; Jastrzębski, Michał K; Karcz, Tadeusz; Olejarz-Maciej, Agnieszka; Sumara, Agata; Laitinen, Tuomo; Wróbel, Tomasz M; Fornal, Emilia; Castro, Marián; Kaczor, Agnieszka A

Development of a novel AAK1 inhibitor via Kinobeads-based screening

利用基于Kinobeads的筛选方法开发新型AAK1抑制剂

Akari Yoshida # ,Satomi Ohtsuka # ,Fumiya Matsumoto ,Tomoyuki Miyagawa ,Rei Okino ,Yumeya Ikeda ,Natsume Tada ,Akira Gotoh ,Masaki Magari ,Naoya Hatano ,Ryo Morishita ,Ayano Satoh ,Yukinari Sunatsuki ,Ulf J Nilsson ,Teruhiko Ishikawa ,Hiroshi Tokumitsu

Recent progress in discovery of novel AAK1 inhibitors: from pain therapy to potential anti-viral agents

新型AAK1抑制剂发现的最新进展:从疼痛治疗到潜在的抗病毒药物

Yuan, Ying-Hui; Mao, Nian-Dong; Duan, Ji-Long; Zhang, Hang; Garrido, Carmen; Lirussi, Frédéric; Gao, Yuan; Xie, Tian; Ye, Xiang-Yang

Evaluating the ability of some natural phenolic acids to target the main protease and AAK1 in SARS COV-2

评估某些天然酚酸靶向SARS-CoV-2主要蛋白酶和AAK1的能力

Ghamry, Heba I; Belal, Amany; El-Ashrey, Mohamed Kandeel; Tawfik, Haytham O; Alsantali, Reem I; Obaidullah, Ahmad J; El-Mansi, Ahmed A; Abdelrahman, Doaa

AAK1-like: A putative pseudokinase with potential roles in cargo uptake in bloodstream form Trypanosoma brucei parasites

AAK1样蛋白:一种假定的假激酶,可能在布氏锥虫血液型寄生虫的货物摄取中发挥作用

Black, Jennifer A; Klinger, Christen M; Lemgruber, Leandro; Dacks, Joel B; Mottram, Jeremy C; McCulloch, Richard

Funnel metadynamics and behavioral studies reveal complex effect of D2AAK1 ligand on anxiety-like processes

漏斗元动力学和行为学研究揭示了D2AAK1配体对焦虑样过程的复杂影响

Bartuzi, Damian; Kędzierska, Ewa; Targowska-Duda, Katarzyna M; Koszła, Oliwia; Wróbel, Tomasz M; Jademyr, Simon; Karcz, Tadeusz; Szczepańska, Katarzyna; Stępnicki, Piotr; Wronikowska-Denysiuk, Olga; Biała, Grażyna; Handzlik, Jadwiga; Kristensen, Jesper L; Poso, Antti; Kaczor, Agnieszka A

Quadruple Target Evaluation of Diversity-Optimized Halogen-Enriched Fragments (HEFLibs) Reveals Substantial Ligand Efficiency for AP2-Associated Protein Kinase 1 (AAK1)

对多样性优化的卤素富集片段(HEFLibs)进行四重靶点评估,揭示了其对 AP2 相关蛋白激酶 1 (AAK1) 的显著配体效率

Dammann, Marcel; Kramer, Markus; Zimmermann, Markus O; Boeckler, Frank M