日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Morphine Tolerance Gated through EZH2-Mediated Suppression of Trpc5 in Spinal GABAergic Interneurons in Male Mice.

吗啡耐受性是通过 EZH2 介导的脊髓 GABA 能中间神经元中 Trpc5 的抑制而实现的。

TRPV2 and TRPC5 are potential targets for astringent phytochemicals

TRPV2 和 TRPC5 是收敛性植物化学物质的潜在靶点。

Kadkova, Anna; Kosinova, Kamila; Klouckova, Marketa; Strachotova, Dita; Barvik, Ivan; Zimova, Lucie; Vlachova, Viktorie

TrpC5 silencing reduces cell invasion and migration and enhances radiosensitivity in papillary thyroid carcinoma cells.

TrpC5 沉默可降低乳头状甲状腺癌细胞的侵袭和迁移能力,并增强其放射敏感性。

Yang Jing, Sang Zijiang, Yang Haibing, Cao Lvzhou, Chen Jinxia, Yang Jiaxin, Gong Rixiang, Li Zhihui, Gong Yanping

Structure-guided design of picomolar-level macrocyclic TRPC5 channel inhibitors with antidepressant activity

结构导向设计具有抗抑郁活性的皮摩尔级大环TRPC5通道抑制剂

Che, Tong; Chen, Yixiang; Cheng, Xinyu; Hu, Han; Wu, Xiaoyun; Zhang, Yuting; Yang, Xiaoqiang; Liu, Yinzhen; Liu, Hui; Nan, Weiwei; Wan, Shuangyan; Yang, Mingxing; Zeng, Bo; Li, Jian; Zhang, Jin; Xiong, Bing

LncRNA NEAT1 contributes to multiple myeloma progression via upregulating ARPC5 by sponging miR-133a.

LncRNA NEAT1 通过海绵吸附 miR-133a 上调 ARPC5,从而促进多发性骨髓瘤的进展。

Wang Fujue, Zeng Piaorong, Lu Zhongwei, Long Xingxing, Luo Cong, Zuo Juan, Cao Yixiong, Wen Feng, Li Junjun, Luo Zeyu

Structural and accessibility studies highlight the differential binding of clemizole to TRPC5 and TRPC6

结构和可及性研究突显了克米唑与TRPC5和TRPC6的差异性结合。

Saqib, Uzma; Demaree, Isaac S; Obukhov, Alexander G; Baig, Mirza S; Khan, Mohd Shahnawaz; Altwaijry, Nojood; Nasution, Mochammad Arfin Fardiansyah; Mizuguchi, Kenji; Hajela, Krishnan

Tricyclic antidepressants dose-dependently modulate the biphasic activity of the TRPC5 channel through opioid receptors

三环类抗抑郁药通过阿片受体以剂量依赖的方式调节TRPC5通道的双相活性。

Jeong, Byeongseok; Chung, Ji Yeon; Jun, Jae Yeoul; Hong, Chansik

N-palmitoyl glycine differentially modulates TRPM4 and TRPC5 and is causally linked to Brugada syndrome

N-棕榈酰甘氨酸对TRPM4和TRPC5具有不同的调节作用,并且与布鲁加达综合征存在因果关系。

Xu, Hongxuan; Li, Bingxun; Chen, Ying; Lin, Yanyun; Zhang, An; Wu, Lin

TRPC5: a new entry to the chromaffin cell's palette of ion channels that control adrenal response to hypoglycemia

TRPC5:嗜铬细胞离子通道家族的新成员,该家族控制着肾上腺对低血糖的反应

Carbone, Emilio

Functional determinants of lysophospholipid- and voltage-dependent regulation of TRPC5 channel

溶血磷脂和电压依赖性 TRPC5 通道调节的功能决定因素

Alexandra Ptakova, Lucie Zimova, Ivan Barvik, Robin S Bon, Viktorie Vlachova