日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction: Hybrid AI/physics pipeline for miniprotein binder prioritization: application to the BRD3 ET domain

更正:用于微型蛋白结合剂优先级排序的混合人工智能/物理流程:应用于 BRD3 ET 结构域

Gaza, Jokent; Roth, Monica J; Montelione, Gaetano T; Perez, Alberto

BRD3 PROTAC degrader targets H3K18ac to alleviate retinal microglia-driven uveitis.

BRD3 PROTAC 降解剂靶向 H3K18ac 以缓解视网膜小胶质细胞驱动的葡萄膜炎。

Zhang Zhi, Lan Tianlong, Liu Yongbo, Yang Hui, Shu Nan, Li Ruonan, Li Wanqian, Zhou Qian, Yang Peizeng, Rao Yu, Hou Shengping

Hybrid AI/physics pipeline for miniprotein binder prioritization: application to the BRD3 ET domain

用于微型蛋白结合剂优先级排序的混合人工智能/物理流程:应用于 BRD3 ET 结构域

Gaza, Jokent; Roth, Monica J; Montelione, Gaetano T; Perez, Alberto

Bromodomain and Extra-Terminal Family Proteins BRD2, BRD3, and BRD4 Contribute to H19-Dependent Transcriptional Regulation of Cell Adhesion Molecules, Modulating Metastatic Dissemination Program in Prostate Cancer

溴结构域和末端外结构域家族蛋白BRD2、BRD3和BRD4参与H19依赖的细胞黏附分子转录调控,从而调节前列腺癌的转移扩散程序。

Valeria Pecci ,Melissa Borsa ,Aurora Aiello ,Sara De Martino ,Luca Cis ,Cristian Ripoli ,Dante Rotili ,Francesco Pierconti ,Francesco Pinto ,Claudio Grassi ,Carlo Gaetano ,Antonella Farsetti ,Simona Nanni

Alkylamine-tethered molecules recruit FBXO22 for targeted protein degradation

烷基胺连接的分子招募FBXO22进行靶向蛋白质降解

Chrysanthi Kagiou ,Jose A Cisneros ,Jakob Farnung ,Joanna Liwocha ,Fabian Offensperger ,Kevin Dong ,Ka Yang ,Gary Tin ,Christina S Horstmann ,Matthias Hinterndorfer ,Joao A Paulo ,Natalie S Scholes ,Juan Sanchez Avila ,Michaela Fellner ,Florian Andersch ,J Thomas Hannich ,Johannes Zuber ,Stefan Kubicek ,Steven P Gygi ,Brenda A Schulman ,Georg E Winter

BRD3308 suppresses macrophage oxidative stress and pyroptosis via upregulating acetylation of H3K27 in sepsis-induced acute lung injury

BRD3308通过上调H3K27乙酰化来抑制脓毒症诱导的急性肺损伤中的巨噬细胞氧化应激和细胞焦亡。

Liu, Bohao; Li, Ning; Liu, Yi; Zhang, Yan; Qu, Limei; Cai, Hongfei; Li, Yang; Wu, Xiaojing; Geng, Qing

Genomic insights from Lactiplantibacillus plantarum BRD3A isolated from Atingba, a traditional fermented rice-based beverage and analysis of its potential for probiotic and antimicrobial activity against Methicillin-resistant Staphylococcus aureus

从传统发酵米酒阿廷巴中分离得到的植物乳杆菌BRD3A的基因组信息及其对耐甲氧西林金黄色葡萄球菌的益生菌和抗菌活性分析

Huidrom, Surmani; Ngashangva, Ng; Khumlianlal, Joshua; Sharma, Kongbrailatpam Chandradev; Mukherjee, Pulok Kumar; Devi, Sarangthem Indira

BRD2 and BRD3 genes independently evolved RNA structures to control unproductive splicing

BRD2和BRD3基因独立进化出RNA结构来控制无效剪接。

Petrova, Marina; Margasyuk, Sergey; Vorobeva, Margarita; Skvortsov, Dmitry; Dontsova, Olga A; Pervouchine, Dmitri D

p300/CBP degradation is required to disable the active AR enhanceosome in prostate cancer

p300/CBP 降解是关闭前列腺癌中活性 AR 增强体所必需的

Jie Luo, Zhixiang Chen, Yuanyuan Qiao, Jean Ching-Yi Tien, Eleanor Young, Rahul Mannan, Somnath Mahapatra, Tongchen He, Sanjana Eyunni, Yuping Zhang, Yang Zheng, Fengyun Su, Xuhong Cao, Rui Wang, Yunhui Cheng, Rithvik Seri, James George, Miriam Shahine, Stephanie J Miner, Ulka Vaishampayan, Mi Wang,

Acetyl-methyllysine marks chromatin at active transcription start sites

乙酰甲基赖氨酸在活性转录起始位点标记染色质

William J Lu-Culligan #, Leah J Connor #, Yixuan Xie, Babatunde E Ekundayo, Brendan T Rose, Martin Machyna, Andreas P Pintado-Urbanc, Joshua T Zimmer, Isaac W Vock, Natarajan V Bhanu, Megan C King, Benjamin A Garcia, Franziska Bleichert, Matthew D Simon