日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dysregulation of the BRD2-FGF17 Signal Pathway Induces Abnormal Forebrain Development Associated with Schizophrenia.

BRD2-FGF17信号通路失调导致与精神分裂症相关的前脑发育异常。

Yu Xiao, Du Jiacheng, Zhou Chenger, Huang Yongheng, Li Huijuan, Cohen Bruce M, Chung Sangmi, Shao Zhicheng

Interaction of coronavirus E protein with BRD2 plays important regulatory roles in viral replication and induction of pro-inflammatory response.

冠状病毒 E 蛋白与 BRD2 的相互作用在病毒复制和诱导促炎反应中起着重要的调控作用。

Li Shumin, Liu Ding Xiang

INO80/SWR remodelers regulate Pol II transcription through BRD2 and chromatin landscape.

INO80/SWR 重塑因子通过 BRD2 和染色质结构调控 Pol II 转录。

Liu Meitong, Xu Qiqin, Wang Hui, Ji Xiong

Overcoming BET-inhibitor JQ1 resistance in aggressive non-small cell lung cancer by inducing ferroptosis via inhibition of the BRD2-FTH1 axis.

通过抑制 BRD2-FTH1 轴诱导铁死亡,克服侵袭性非小细胞肺癌中 BET 抑制剂 JQ1 的耐药性。

Scicchitano Stefania, Garofalo Cinzia, Stella Beatrice, Santamaria Gianluca, Cozzolino Flora, Monaco Vittoria, Biamonte Flavia, Monti Maria, Vecchio Eleonora, Faniello Maria Concetta

BRD2 phase separation activates super-enhancer-driven ATG7 transcription to promote ferritinophagy in depression.

BRD2 相分离激活超级增强子驱动的 ATG7 转录,从而促进抑郁症中的铁蛋白自噬。

Targeting of vulnerabilities of drug-tolerant persisters identified through functional genetics delays tumor relapse

通过功能遗传学鉴定的耐药持久细胞的脆弱性可以延缓肿瘤复发

Mengnuo Chen, Sara Mainardi, Cor Lieftink, Arno Velds, Iris de Rink, Chen Yang, Hendrik J Kuiken, Ben Morris, Finn Edwards, Fleur Jochems, Olaf van Tellingen, Manon Boeije, Natalie Proost, Robin A Jansen, Shifan Qin, Haojie Jin, J C Koen van der Mijn, Arnout Schepers, Subramanian Venkatesan, Wenxin

Functional E3 ligase hotspots and resistance mechanisms to small-molecule degraders

功能性E3连接酶热点及对小分子降解剂的耐药机制

Alexander Hanzl ,Ryan Casement # ,Hana Imrichova # ,Scott J Hughes ,Eleonora Barone ,Andrea Testa ,Sophie Bauer ,Jane Wright ,Matthias Brand ,Alessio Ciulli ,Georg E Winter

Exploring the target scope of KEAP1 E3 ligase-based PROTACs

探索基于 KEAP1 E3 连接酶的 PROTAC 的靶标范围

Guangyan Du, Jie Jiang, Nathaniel J Henning, Nozhat Safaee, Eriko Koide, Radosław P Nowak, Katherine A Donovan, Hojong Yoon, Inchul You, Hong Yue, Nicholas A Eleuteri, Zhixiang He, Zhengnian Li, Hubert T Huang, Jianwei Che, Behnam Nabet, Tinghu Zhang, Eric S Fischer, Nathanael S Gray

Targeting BET Proteins With a PROTAC Molecule Elicits Potent Anticancer Activity in HCC Cells

利用PROTAC分子靶向BET蛋白可诱导HCC细胞产生强效抗癌活性

Huapeng Zhang ,Gongquan Li ,Yi Zhang ,Jihua Shi ,Bing Yan ,Hongwei Tang ,Sanyang Chen ,Jiakai Zhang ,Peihao Wen ,Zhihui Wang ,Chun Pang ,Jie Li ,Wenzhi Guo ,Shuijun Zhang

Brd2 haploinsufficiency extends lifespan and healthspan in C57B6/J mice

Brd2单倍体不足延长了C57B6/J小鼠的寿命和健康寿命

Pathak, Shilpa; Stewart, William C L; Burd, Christin E; Hester, Mark E; Greenberg, David A