日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cucurbitacin B inhibits HIF-1α and attenuates non-small cell lung cancer via ZFP91

葫芦素B通过ZFP91抑制HIF-1α并减弱非小细胞肺癌

Lei Song #,Jing Han #,Run Wang #,Shen Cao,Yi Tai,Xinyu Wang,Yanjin Zheng,Shufeng Jin,Yue Xing,Hong Xiang Zuo,Ming Yue Li,Juan Ma,Xuejun Jin

Correction: Cucurbitacin B inhibits HIF-1α and attenuates non-small cell lung cancer via ZFP91

更正:葫芦素B通过ZFP91抑制HIF-1α并减弱非小细胞肺癌

Song, Lei; Han, Jing; Wang, Run; Cao, Shen; Tai, Yi; Wang, Xinyu; Zheng, Yanjin; Jin, Shufeng; Xing, Yue; Zuo, Hong Xiang; Li, Ming Yue; Ma, Juan; Jin, Xuejun

Proteolysis-targeting chimeras with reduced off-targets

靶向蛋白水解的嵌合体,脱靶率较低

Tuan M Nguyen #, Vedagopuram Sreekanth #, Arghya Deb #, Praveen Kokkonda #, Praveen K Tiwari, Katherine A Donovan, Veronika Shoba, Santosh K Chaudhary, Jaron A M Mercer, Sophia Lai, Ananthan Sadagopan, Max Jan, Eric S Fischer, David R Liu, Benjamin L Ebert, Amit Choudhary

Lenalidomide derivatives and proteolysis-targeting chimeras for controlling neosubstrate degradation

来那度胺衍生物和靶向蛋白水解的嵌合体用于控制新底物降解

Satoshi Yamanaka,Hirotake Furihata,Yuta Yanagihara,Akihito Taya,Takato Nagasaka,Mai Usui,Koya Nagaoka,Yuki Shoya,Kohei Nishino,Shuhei Yoshida,Hidetaka Kosako,Masaru Tanokura,Takuya Miyakawa,Yuuki Imai,Norio Shibata,Tatsuya Sawasaki

ZFP91 disturbs metabolic fitness and antitumor activity of tumor-infiltrating T cells

ZFP91 干扰肿瘤浸润 T 细胞的代谢适应性和抗肿瘤活性

Feixiang Wang, Yuerong Zhang, Xiaoyan Yu, Xiao-Lu Teng, Rui Ding, Zhilin Hu, Aiting Wang, Zhengting Wang, Youqiong Ye, Qiang Zou

Discovery of a Napabucasin PROTAC as an Effective Degrader of the E3 Ligase ZFP91

发现 Napabucasin PROTAC 是 E3 连接酶 ZFP91 的有效降解剂

Maha Hanafi, Xinde Chen, Nouri Neamati

E3 ligase ZFP91 inhibits Hepatocellular Carcinoma Metabolism Reprogramming by regulating PKM splicing

E3连接酶ZFP91通过调控PKM剪接抑制肝细胞癌代谢重编程

De Chen,Yanjie Wang,Ruixun Lu,Xiaofeng Jiang,Xinhui Chen,Nan Meng,Min Chen,Shan Xie,Guang-Rong Yan

IMiDs induce FAM83F degradation via an interaction with CK1α to attenuate Wnt signalling

IMiD 通过与 CK1α 相互作用诱导 FAM83F 降解,从而减弱 Wnt 信号传导

Karen Dunbar, Thomas J Macartney, Gopal P Sapkota

Defining the human C2H2 zinc finger degrome targeted by thalidomide analogs through CRBN

通过 CRBN 定义沙利度胺类似物靶向的人类 C2H2 锌指降解组

Quinlan L Sievers, Georg Petzold, Richard D Bunker, Aline Renneville, Mikołaj Słabicki, Brian J Liddicoat, Wassim Abdulrahman, Tarjei Mikkelsen, Benjamin L Ebert, Nicolas H Thomä

Crbn I391V is sufficient to confer in vivo sensitivity to thalidomide and its derivatives in mice

Crbn I391V 足以使小鼠对沙利度胺及其衍生物产生体内敏感性

Emma C Fink, Marie McConkey, Dylan N Adams, Saurav D Haldar, James A Kennedy, Andrew A Guirguis, Namrata D Udeshi, D R Mani, Michelle Chen, Brian Liddicoat, Tanya Svinkina, Andrew T Nguyen, Steven A Carr, Benjamin L Ebert