日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Deubiquitinase USP37 enhances the anti-HIV-2/SIV ability of the host restriction factor SAMHD1

去泛素化酶USP37增强宿主限制因子SAMHD1的抗HIV-2/SIV能力

Wenzhe Cui ,Hongfei Wang ,Yuan Gao ,Xue Zhang ,Jingguo Xin ,Zhaolong Li ,Guangquan Li ,Wenying Gao ,Wenyan Zhang

Inhibitors of SAMHD1 Obtained from Chemical Tethering to the Guanine Antiviral Acyclovir

通过化学方法将抗病毒药物阿昔洛韦连接到鸟嘌呤上而获得的SAMHD1抑制剂

Matthew Egleston ,Shridhar Bhat ,A Hasan Howlader ,Mario A Bianchet ,Yi Liu ,Laura Maria Lopez Rovira ,Brandon Smith ,Marc M Greenberg ,James T Stivers

ssDNA and ssRNA Promote Phase Condensation of SAMHD1

单链DNA和单链RNA促进SAMHD1的相凝聚

Brandon E Smith ,Ankita Pohnerkar ,Benjamin Orris ,Shridhar Bhat ,Matthew Egleston ,James T Stivers

Identification and evaluation of small-molecule inhibitors against the dNTPase SAMHD1 via a comprehensive screening funnel

通过综合筛选流程鉴定和评价针对 dNTPase SAMHD1 的小分子抑制剂

Si Min Zhang ,Cynthia B J Paulin ,Huazhang Shu ,Miriam Yagüe-Capilla ,Maurice Michel ,Petra Marttila ,Florian Ortis ,Henri Colyn Bwanika ,Christopher Dirks ,Rajagopal Papagudi Venkatram ,Elisée Wiita ,Ann-Sofie Jemth ,Ingrid Almlöf ,Olga Loseva ,Femke M Hormann ,Tobias Koolmeister ,Erika Linde ,Sun Lee ,Sabin Llona-Minguez ,Martin Haraldsson ,Hanna Axelsson ,Kia Strömberg ,Evert J Homan ,Martin Scobie ,Thomas Lundbäck ,Thomas Helleday ,Sean G Rudd

Preclinical Evaluation of Soluble Epoxide Hydrolase Inhibitor AMHDU against Neuropathic Pain

可溶性环氧化物水解酶抑制剂AMHDU治疗神经性疼痛的临床前评价

Denis Babkov ,Natalya Eliseeva ,Kristina Adzhienko ,Viktoria Bagmetova ,Dmitry Danilov ,Cynthia B McReynolds ,Christophe Morisseau ,Bruce D Hammock ,Vladimir Burmistrov

Guanine-containing ssDNA and RNA induce dimeric and tetrameric structural forms of SAMHD1

含鸟嘌呤的单链DNA和RNA诱导SAMHD1形成二聚体和四聚体结构形式。

Benjamin Orris ,Min Woo Sung ,Shridhar Bhat ,Yingrong Xu ,Kevin W Huynh ,Seungil Han ,Darren C Johnson ,Benedikt Bosbach ,David J Shields ,James T Stivers

Deficiency for SAMHD1 activates MDA5 in a cGAS/STING-dependent manner

SAMHD1 的缺乏以 cGAS/STING 依赖的方式激活 MDA5。

Tina Schumann ,Santiago Costas Ramon ,Nadja Schubert ,Mohamad Aref Mayo ,Melanie Hega ,Katharina Isabell Maser ,Servi-Remzi Ada ,Lukas Sydow ,Mona Hajikazemi ,Markus Badstübner ,Patrick Müller ,Yan Ge ,Farhad Shakeri ,Andreas Buness ,Benjamin Rupf ,Stefan Lienenklaus ,Barbara Utess ,Lina Muhandes ,Michael Haase ,Luise Rupp ,Marc Schmitz ,Thomas Gramberg ,Nicolas Manel ,Gunther Hartmann ,Thomas Zillinger ,Hiroki Kato ,Stefan Bauer ,Alexander Gerbaulet ,Katrin Paeschke ,Axel Roers ,Rayk Behrendt

SAMHD1 deacetylation by SIRT1 promotes DNA end resection by facilitating DNA binding at double-strand breaks

SIRT1 对 SAMHD1 的去乙酰化作用通过促进 DNA 与双链断裂处的结合来促进 DNA 末端切除。

Priya Kapoor-Vazirani ,Sandip K Rath ,Xu Liu ,Zhen Shu ,Nicole E Bowen ,Yitong Chen ,Ramona Haji-Seyed-Javadi ,Waaqo Daddacha ,Elizabeth V Minten ,Diana Danelia ,Daniela Farchi ,Duc M Duong ,Nicholas T Seyfried ,Xingming Deng ,Eric A Ortlund ,Baek Kim ,David S Yu

Equine lentivirus counteracts SAMHD1 restriction by Rev-mediated degradation of SAMHD1 via the BECN1-dependent lysosomal pathway

马慢病毒通过 BECN1 依赖的溶酶体途径,利用 Rev 介导的 SAMHD1 降解来对抗 SAMHD1 的限制作用。

Huiling Ren,Xin Yin,Chao Su,Miaomiao Guo,Xue-Feng Wang,Lei Na,Yuezhi Lin,Xiaojun Wang

TRAF6 and TAK1 Contribute to SAMHD1-Mediated Negative Regulation of NF-κB Signaling

TRAF6 和 TAK1 参与 SAMHD1 介导的 NF-κB 信号负调控

Constanza E Espada # ,Corine St Gelais # ,Serena Bonifati # ,Victoria V Maksimova ,Michael P Cahill ,Sun Hee Kim ,Li Wu