日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Cyclin C-CDK8/19 Mediator kinase module controls PRCC-TFE3 driven senescence in renal epithelium and tumorigenesis in TFE3-RCC

细胞周期蛋白C-CDK8/19介导激酶模块控制PRCC-TFE3驱动的肾上皮细胞衰老和TFE3-RCC的肿瘤发生。

Kuroda, Shoichiro; Funasaki, Shintaro; Nishizawa, Hidekazu; Schmidt, Laura S; Kurahashi, Ryoma; Ito, Takaaki; Arima, Yuichiro; Tanaka, Miwa; Kitada, Atsuya; James, Amy M; Hasumi, Hisashi; Jikuya, Ryosuke; Makiyama, Kazuhide; Kurotaki, Daisuke; Minami, Takashi; Difilippantonio, Simone; Linehan, W Marston; Oike, Yuichi; Sawa, Tomohiro; Tanaka, Yasuhito; Suda, Toshio; Yokokawa, Ryuji; Nakamura, Takuro; Baba, Masaya; Kamba, Tomomi

Inhibition of CDK8 rescues impaired ischemic fracture healing

抑制 CDK8 可挽救缺血性骨折愈合受损。

Capobianco, Christina A; Song, Michelle J; Farrell, Easton C; Knights, Alexander J; Kessell, Karen; Donneys, Alexis; Schmanski, Jeanna T; Schroeder, Luke R; Chen, Mengqian; Roninson, Igor B; Wagley, Yadav; Maerz, Tristan; Hankenson, Kurt D

Anoikis resistance and metastasis of ovarian cancer can be overcome by CDK8/19 mediator kinase inhibition

CDK8/19介导激酶抑制可以克服卵巢癌的抗凋亡和转移。

Monavarian, Mehri; Rajkarnikar, Resha; Page, Emily Faith; Kumari, Asha; Quintero Macias, Liz; Massicano, Felipe; Lee, Nam Y; Sahoo, Sarthak; Hempel, Nadine; Jolly, Mohit Kumar; Ianov, Lara; Worthey, Elizabeth; Singh, Abhyudai; Roninson, Igor B; Broude, Eugenia V; Chen, Mengqian; Mythreye, Karthikeyan

Runx2 acetylation enhances pulmonary inflammation in chronic obstructive pulmonary disease through activating CDK8.

Runx2 乙酰化通过激活 CDK8 增强慢性阻塞性肺病中的肺部炎症。

Ma Yi-Cheng, Chen Dan-Lei, Wu Ju-Hong, Tang Fei, Sui Tian-Rui, Wu Zhi-Yong, He Qi-Yuan, Wang Yu, Tang Min-Min, Hua Dong-Xu, Yang Jing, Zhao Hui, Fei Jun, Cao Wei, Fu Lin

CDK8 Inhibition Increases E2F1 Transcriptional Activity and Promotes STAT3-Dependent Suppression of Mcl-1 in Triple-Negative Breast Cancer Cell Line MDA-MB-468

CDK8抑制可增强E2F1转录活性,并促进STAT3依赖性抑制三阴性乳腺癌细胞系MDA-MB-468中的Mcl-1表达。

Do, Sandra; Li, Shengxi; Xiong, Rui; Spear, Jensen M; Lu, Zhixin; Chan, William K; Russu, Wade A

Abnormal circ-CDK8 expression affects periodontitis development by regulating let-7b-5p/MAP4K3 signaling

circ-CDK8表达异常通过调节let-7b-5p/MAP4K3信号通路影响牙周炎的发展

Li, Yabo; Yang, Cailing; Jin, Mengdie; Liu, Ting; Yuan, Changqing; Zheng, Jingjing

Therapeutic potential of CDK8 inhibitor combined with sorafenib for hepatocellular carcinoma: mechanistic insights and in vitro validation

CDK8抑制剂联合索拉非尼治疗肝细胞癌的潜力:机制研究及体外验证

Gao, Li; Wu, Hong; Du, Sheng-Yuan; Lv, Zi-Li

let-7c-5p promotes fracture healing by downregulating CDK8.

let-7c-5p 通过下调 CDK8 促进骨折愈合。

Liu Wei, Zhang Jinxiang, Chen Xi, Cheng Bin, Li Qiang, Li Lin, Yang Hongbin

Impact of MED12 mutation and CDK8 activity on uterine leiomyoma growth and response to gonadotropin-releasing hormone agonist treatment.

MED12 突变和 CDK8 活性对子宫平滑肌瘤生长及促性腺激素释放激素激动剂治疗反应的影响。

Tanioka Saki, Asano Ryoko, Ota Yukihide, Nagai Koichi, Takenaka Katsuya, Mizushima Taichi, Miyagi Yohei, Miyagi Etsuko

Romaciclib, a CDK8/CDK19 inhibitor, can overcome venetoclax resistance through a combinatorial strategy

罗玛西利(Romaciclib)是一种 CDK8/CDK19 抑制剂,可通过联合治疗策略克服维奈托克耐药性。

Pakulska, Urszula; Obacz, Marta; Woźnicki, Jerzy; Wiklik, Katarzyna; Chakraborty, Samarpana; Micek, Marta; Mohanty, Vakul; Coelho, Diego; Adamczyk, Elżbieta; Gołas, Aniela; Moszyńska, Adrianna; Zhang, Hui; Cybulska-Lubak, Magdalena; Kaniuga, Ewelina; Sandowska-Markiewicz, Zuzanna; Konopleva, Marina; Mikula, Michał; Juszczyński, Przemysław; Shastri, Aditi; Baran, Natalia; Rzymski, Tomasz; Mazan, Milena