Helicobacter pylori CagA inhibits PAR1-MARK family kinases by mimicking host substrates

幽门螺杆菌CagA通过模拟宿主底物抑制PAR1-MARK家族激酶

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Abstract

The CagA protein of Helicobacter pylori interacts with numerous cellular factors and is associated with increased virulence and risk of gastric carcinoma. We present here the cocrystal structure of a subdomain of CagA with the human kinase PAR1b/MARK2, revealing that a CagA peptide mimics substrates of this kinase family, resembling eukaryotic protein kinase inhibitors. Mutagenesis of conserved residues central to this interaction renders CagA inactive as an inhibitor of MARK2.

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