Enhancing k(cat) prediction through residue-aware attention mechanism and pre-trained representations

通过残差感知注意力机制和预训练表征增强k(cat)预测

阅读:1

Abstract

The turnover number (k(cat)) is a key parameter in enzyme kinetics that quantifies catalytic efficiency and underpins mechanistic understanding of enzyme activity. However, existing computational approaches for k(cat) prediction often suffer from limited accuracy and generalization, largely because most models rely only on substrate information and neglect the role of the full reaction context. Although TurNuP partially addresses this limitation by encoding entire reactions using binary fingerprints, its two-stage design separates enzyme and reaction modeling, limiting both predictive performance and interpretability. Here, we present PMAK, a deep learning framework that integrates pre-trained representations of enzyme sequences and reaction SMILES with a residue-aware attention mechanism. By jointly modeling enzymes and reactions, PMAK captures their interactions and highlights key residues contributing to catalytic activity. Comprehensive evaluations demonstrate that PMAK consistently outperforms existing methods, achieving average R(2) improvements of approximately 16.9% and 10.0% over TurNuP under new-reaction and new-enzyme settings, respectively, in five-fold cross-validation. Beyond improved accuracy, PMAK provides interpretable insights into residues associated with enzyme catalysis, offering a robust and informative tool for enzyme kinetic prediction and related applications.

特别声明

1、本页面内容包含部分的内容是基于公开信息的合理引用;引用内容仅为补充信息,不代表本站立场。

2、若认为本页面引用内容涉及侵权,请及时与本站联系,我们将第一时间处理。

3、其他媒体/个人如需使用本页面原创内容,需注明“来源:[生知库]”并获得授权;使用引用内容的,需自行联系原作者获得许可。

4、投稿及合作请联系:info@biocloudy.com。