Mechanism of astaxanthin improving exercise-induced muscle damage: an integrated approach using network pharmacology, molecular dynamics simulation, and experimental validation

虾青素改善运动性肌肉损伤的机制:一种结合网络药理学、分子动力学模拟和实验验证的综合方法

阅读:1

Abstract

This research evaluated the potential mechanisms of ASX on EIMD. The network pharmacology, machine learning, and transcription sequencing were applied to explore the targets of ASX improving EIMD, which were then validated by molecular dynamics simulation and experiments. Twenty five key targets were screened after topological network analysis and mainly enriched in the Toll-like receptor signaling pathway, NF-κB signaling pathway, and Cytokine-cytokine receptor interaction. Through machine learning algorithms, four candidate targets, including CCL2, NFE2L2, TLR4, and TGFB1, were acquired. Combined with transcriptome sequencing results, CCL2 and TLR4 were finally identified as core targets for ASX to improve EIMD. Molecular dynamics simulation confirmed the strong binding affinity of ASX-CCL2 and ASX-TLR4 complexes. Besides, RT-PCR and Western blot revealed that the mRNA and protein expression of the TLR4/MyD88/NF-κB/CCL2/CCR2 pathway in the EIMD model were significantly down-regulated after ASX intervention. ASX might effectively attenuate muscle damage during exercise through the TLR4/MyD88/NF-κB/CCL2/CCR2 pathway. SUPPLEMENTARY INFORMATION: The online version contains supplementary material available at 10.1007/s10068-026-02086-z.

特别声明

1、本页面内容包含部分的内容是基于公开信息的合理引用;引用内容仅为补充信息,不代表本站立场。

2、若认为本页面引用内容涉及侵权,请及时与本站联系,我们将第一时间处理。

3、其他媒体/个人如需使用本页面原创内容,需注明“来源:[生知库]”并获得授权;使用引用内容的,需自行联系原作者获得许可。

4、投稿及合作请联系:info@biocloudy.com。