Hybrids of Layered Double Hydroxides and Sodium Dodecyl Sulfate: Structural Effects on the Controlled Release of Pretilachlor

层状双氢氧化物与十二烷基硫酸钠的杂化物:结构对吡草胺控释的影响

阅读:1

Abstract

Organo-layered double hydroxides (OLDHs) are widely used as slow-release carriers for drugs but are rarely used in controlled drug release. To develop slow-release substrates of pretilachlor with excellent controlled release properties, OLDH hybrids were prepared by intercalating different masses of sodium dodecyl sulfate (SDS) into MgAl-LDHs. The underlying structural characteristics were analyzed by X-ray diffraction (XRD), Fourier Transform Infrared Spectroscopy (FT-IR), scanning electron microscopy (SEM), and contact angle measurements. Also, the adsorption capacity and release properties of OLDHs were explored by batch adsorption isotherms, adsorption kinetics, and release kinetics to reveal the structural effects of OLDHs on the release of pretilachlor. The results showed that the release of pretilachlor from OLDHs was dominated by Fickian diffusion and was closely related to the adsorption capacity and permeability of the matrix. The intercalation of SDS enhanced the hydrophobicity of LDHs, resulting in a higher adsorption capacity for pretilachlor and a lower permeability. Furthermore, as the SDS loading amount increased from 0.5 to 4.0 g, the adsorption capacity of the OLDHs was further enhanced (k (F) value increased from 2.52 to 12.83), while the permeability (d (001)/f (oc) value) reversed, decreasing from 0.21 to 0.09. The release kinetics demonstrated that the release rate of pretilachlor from OLDHs was significantly lower compared to pure LDHs and showed a continuous decrease with increasing SDS loading amounts. The release time of 50% (T (50)) pretilachlor from OLDHs with SDS loading amounts of 25%, 50%, 100%, and 200% of the anion exchange capacity was 4.78, 8.28, 25.4, and 45.34 times longer than the release time from pure LDHs. This displayed a strong curvilinear relationship with the adsorption rate constant k (F) and permeability d (001)/f (oc) and a good linear relationship with the added amount of SDS. These findings highlight the potential of OLDHs in preparing pretilachlor controlled release formulations.

特别声明

1、本页面内容包含部分的内容是基于公开信息的合理引用;引用内容仅为补充信息,不代表本站立场。

2、若认为本页面引用内容涉及侵权,请及时与本站联系,我们将第一时间处理。

3、其他媒体/个人如需使用本页面原创内容,需注明“来源:[生知库]”并获得授权;使用引用内容的,需自行联系原作者获得许可。

4、投稿及合作请联系:info@biocloudy.com。