日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Hyperactive Signalosome in Acute Myeloid Leukemia Drives Addiction to a Tumor-Specific Hsp90 Species

急性髓系白血病中过度活跃的信号体导致对肿瘤特异性 Hsp90 物种的成瘾

Hongliang Zong, Alexander Gozman, Eloisi Caldas-Lopes, Tony Taldone, Eric Sturgill, Sarah Brennan, Stefan O Ochiana, Erica M Gomes-DaGama, Siddhartha Sen, Anna Rodina, John Koren 3rd, Michael W Becker, Charles M Rudin, Ari Melnick, Ross L Levine, Gail J Roboz, Stephen D Nimer, Gabriela Chiosis, Moni

Heat shock protein 70 inhibitors. 2. 2,5'-thiodipyrimidines, 5-(phenylthio)pyrimidines, 2-(pyridin-3-ylthio)pyrimidines, and 3-(phenylthio)pyridines as reversible binders to an allosteric site on heat shock protein 70

热休克蛋白 70 抑制剂。2. 2,5'-硫代二嘧啶、5-(苯硫基)嘧啶、2-(吡啶-3-基硫基)嘧啶和 3-(苯硫基)吡啶作为热休克蛋白 70 变构位点的可逆结合剂

Tony Taldone, Yanlong Kang, Hardik J Patel, Maulik R Patel, Pallav D Patel, Anna Rodina, Yogita Patel, Alexander Gozman, Ronnie Maharaj, Cristina C Clement, Alvin Lu, Jason C Young, Gabriela Chiosis

Heat shock protein 70 inhibitors. 1. 2,5'-thiodipyrimidine and 5-(phenylthio)pyrimidine acrylamides as irreversible binders to an allosteric site on heat shock protein 70

热休克蛋白 70 抑制剂。1. 2,5'-硫代二嘧啶和 5-(苯硫基)嘧啶丙烯酰胺作为热休克蛋白 70 变构位点的不可逆结合剂

Yanlong Kang, Tony Taldone, Hardik J Patel, Pallav D Patel, Anna Rodina, Alexander Gozman, Ronnie Maharaj, Cristina C Clement, Maulik R Patel, Jeffrey L Brodsky, Jason C Young, Gabriela Chiosis

Affinity purification probes of potential use to investigate the endogenous Hsp70 interactome in cancer

亲和纯化探针可用于研究癌症中的内源性 Hsp70 相互作用组

Anna Rodina, Tony Taldone, Yanlong Kang, Pallav D Patel, John Koren 3rd, Pengrong Yan, Erica M DaGama Gomes, Chenghua Yang, Maulik R Patel, Liza Shrestha, Stefan O Ochiana, Cristina Santarossa, Ronnie Maharaj, Alexander Gozman, Marc B Cox, Hediye Erdjument-Bromage, Ronald C Hendrickson, Leandro Cerc