A novel cell-permeable, selective, and noncompetitive inhibitor of KAT3 histone acetyltransferases from a combined molecular pruning/classical isosterism approach
一种新型的细胞通透性、选择性、非竞争性的 KAT3 组蛋白乙酰转移酶抑制剂,通过分子修剪/经典电子等排方法合成
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm5019687
Ciro Milite, Alessandra Feoli, Kazuki Sasaki, Valeria La Pietra, Amodio Luca Balzano, Luciana Marinelli, Antonello Mai, Ettore Novellino, Sabrina Castellano, Alessandra Tosco, Gianluca Sbardella