日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

AI-Enhanced Adaptive Virtual Screening Platform Enabling Exploration of 69 Billion Molecules Discovers Structurally Validated FSP1 Inhibitors

AI增强型自适应虚拟筛选平台可探索690亿个分子,并发现结构验证的FSP1抑制剂

Cecchini, Domiziana; Nigam, AkshatKumar; Tang, Ming; Reis, Joana; Koop, Matt; Gottinger, Andrea; Nicoll, Callum Robert; Wang, Yao; Jayaraj, Abhilash; Çınaroğlu, Süleyman Selim; Törner, Ricarda; Malets, Yehor; Gehev, Minko; Das, Krishna M Padmanabha; Churion, Kelly; Kim, Jongwan; Thomas, Nidhin; Li, Yong; Seo, Hyuk-Soo; Dhe-Paganon, Sirano; Secker, Christopher; Haddadnia, Mohammad; Hasson, Alexander; Li, Minkai; Kumar, Abhishek; Levin-Konigsberg, Roni; Choi, Eun-Bee; Shapiro, Geoffrey I; Cox, Huel; Sebastian, Luke; Braithwaite, Chelsea; Bashyal, Puspalata; Radchenko, Dmytro S; Kumar, Aditya; Yang, Lei; Aquilanti, Pierre-Yves; Gabb, Henry; Alhossary, Amr; Wagner, Gerhard; Aspuru-Guzik, Alán; Moroz, Yurii S; Kalodimos, Charalampos G; Fackeldey, Konstantin; Schuetz, John D; Mattevi, Andrea; Arthanari, Haribabu; Gorgulla, Christoph

Leveraging relaxation-optimized (1)H-(13)C(F) correlations in 4-(19)F-phenylalanine as atomic beacons for probing structure and dynamics of large proteins

利用4-(19)F-苯丙氨酸中弛豫优化的(1)H-(13)C(F)相关性作为原子信标来探测大型蛋白质的结构和动力学

Boeszoermenyi, Andras; Radeva, Denitsa L; Schindler, Sebastian; Valadares, Veronica; Padmanabha Das, Krishna M; Dubey, Abhinav; Viennet, Thibault; Schmitt, Max; Kast, Peter; Gelev, Vladimir M; Stoyanov, Nikolay; Burdzhiev, Nikola; Petrov, Ognyan; Ficarro, Scott; Marto, Jarred; Geffken, Ezekiel A; Dhe-Paganon, Sirano; Seo, Hyuk-Soo; Alexander, Nathan D; Cooley, Richard B; Mehl, Ryan A; Kovacs, Helena; Anklin, Clemens; Bermel, Wolfgang; Kuprov, Ilya; Takeuchi, Koh; Arthanari, Haribabu

Biophysical and Structural Features of αβT-Cell Receptor Mechanosensing: A Paradigmatic Shift in Understanding T-Cell Activation

αβT细胞受体机械感知的生物物理和结构特征:理解T细胞活化的范式转变

Mallis, Robert J; Brazin, Kristine N; Duke-Cohan, Jonathan S; Akitsu, Aoi; Stephens, Hanna M; Chang-Gonzalez, Ana C; Masi, Daniel J; Kirkpatrick, Evan H; Holliday, Elizabeth L; Feng, Yinnian; Zienkiewicz, Katarzyna J; Lee, Jonathan J; Cinella, Vincenzo; Uberoy, Kaveri I; Tan, Kemin; Wagner, Gerhard; Arthanari, Haribabu; Hwang, Wonmuk; Lang, Matthew J; Reinherz, Ellis L

Targeting transcription factors through an IMiD independent zinc finger domain.

通过不依赖于IMiD的锌指结构域靶向转录因子

Liu Bee Hui, Liu Miao, Radhakrishnan Sridhar, Dai Meng-Yuan, Jaladanki Chaitanya Kumar, Gao Chong, Tang Jing Ping, Kumari Kalpana, Go Mei Lin, Vu Kim Anh L, Kwon Junsu, Seo Hyuk-Soo, Song Kijun, Tian Xi, Feng Li, Tan Justin L, Melkonian Arek V, Liu Zhaoji, Wulf Gerburg, Arthanari Haribabu, Qi Jun, Dhe-Paganon Sirano, Clohessy John G, Choong Yeu Khai, Sivaraman J, Fan Hao, Tenen Daniel G, Chai Li

Dynamic sampling of a surveillance state enables DNA proofreading by Cas9.

通过动态采样监控状态,Cas9 可以进行 DNA 校对

De Paula Viviane S, Dubey Abhinav, Arthanari Haribabu, Sgourakis Nikolaos G

FoxP3 forms a head-to-head dimer in vivo and stabilizes its multimerization on adjacent microsatellites.

FoxP3 在体内形成头对头二聚体,并稳定其在相邻微卫星上的多聚化。

Leng Fangwei, Clark Ryan, Zhang Wenxiang, Viennet Thibault, Wang Cuidie, Arthanari Haribabu, Wang Xi, Hur Sun

Inhibition of dimeric SARS-CoV-2 Mpro displays positive cooperativity and a mixture of covalent and non-covalent binding.

二聚体 SARS-CoV-2 Mpro 的抑制表现出正协同性,并且是共价和非共价结合的混合

Padmanabha Das Krishna M, Chen Jun, Charifson Paul S, Green Jeremy, Tang Henry, Panchal Sanjay, Pu Fan, Korepanova Alla, Dubey Abhinav, Afanador Gustavo, Stojkovic Vladimir, Nocek Boguslaw, Bigelow Lance, Stubbs Sarah H, Davey Robert A, DeGoey David A, Arthanari Haribabu, Namchuk Mark N

Efficacy & safety of high-dose rifampicin in pulmonary tuberculosis: A systematic review & meta-analysis

高剂量利福平治疗肺结核的疗效和安全性:系统评价和荟萃分析

Kannabiran, Bhavani Perumal; Arthanari, Jayanthi; Bhaskar, Adhin; Narayanan, Mukesh Kumar Sathya; Inbaraj, Leeberk Raja

Advanced Imaging Techniques (PET, fMRI, DTI) in Early Detection of Neurodegenerative Diseases: A Systematic Review

先进影像技术(PET、fMRI、DTI)在神经退行性疾病早期检测中的应用:系统评价

Chandrasekar, Santosh Kishor; Arthanari, Jayanthi; Chandrasekar, Kiran Kishor; Gaviria, Elizabeth; Shashank, Singam; Jethi, Achint; John, Jobby; Bopparaju, Sahana; Potulapati, Indra; Mateen, Mohammed Abdul; Hussin, Omniat Amir

Internet Gaming Disorder - An Emerging Digital Epidemic: Exploratory Analysis of Prevalence and Correlates among Young Adults of Tamil Nadu

网络游戏成瘾——一种新兴的数字流行病:对泰米尔纳德邦青年人群患病率及其相关因素的探索性分析

Arthanari, Sakthivel; Geethanjali, S; Hemamalini, B B; Khalique, Najam