日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Novel Human Constitutive Androstane Receptor Agonists with the Imidazo[1,2- a]pyridine Structure

发现具有咪唑并[1,2-a]吡啶结构的新型人类组成型雄烷受体激动剂

Ivana Mejdrová, Jan Dušek, Kryštof Škach, Alžbeta Stefela, Josef Skoda, Karel Chalupský, Klára Dohnalová, Ivona Pavkova, Thales Kronenberger, Azam Rashidian, Lucie Smutná, Vojtěch Duchoslav, Tomas Smutny, Petr Pávek, Radim Nencka

Target Hopping from Protein Kinases to PXR: Identification of Small-Molecule Protein Kinase Inhibitors as Selective Modulators of Pregnane X Receptor from TüKIC Library

从蛋白激酶到PXR的靶点跃迁:从TüKIC库中鉴定出选择性调节孕烷X受体的小分子蛋白激酶抑制剂

Enni-Kaisa Mustonen,Tatu Pantsar,Azam Rashidian,Juliander Reiner,Matthias Schwab,Stefan Laufer,Oliver Burk

Discrepancy in interactions and conformational dynamics of pregnane X receptor (PXR) bound to an agonist and a novel competitive antagonist

孕烷 X 受体 (PXR) 与激动剂和新型竞争性拮抗剂结合的相互作用和构象动力学差异

Azam Rashidian, Enni-Kaisa Mustonen, Thales Kronenberger, Matthias Schwab, Oliver Burk, Stefan A Laufer, Tatu Pantsar