日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Arylhydrazines: Convenient Homogeneous Reductants for Scalable Cross-Coupling

芳基肼:用于可扩展交叉偶联的便捷均相还原剂

Kurig, Nils; Cagan, David A; Harper, Kaid C; Kawamata, Yu; Blackmond, Donna G; Baran, Phil S

Decoding the Nested, Multicycle Mechanism of Ni-Catalyzed Redox-Neutral Cross-Coupling through Temperature Scanning Reaction Calorimetry

通过温度扫描反应量热法解析镍催化氧化还原中性交叉偶联反应的嵌套多循环机理

Cagan, David A; Péter, Áron; Vokits, Benjamin P; Chan, Michael; Baran, Phil S; Blackmond, Donna G

Scalable total synthesis of saxitoxin and related natural products

可规模化合成石房蛤毒素及相关天然产物

Guo, Yinliang; Li, Yiheng; Chen, Sihan; Wu, Yige; Poll, Oscar; Ren, Zhouyang; Liu, Zhonglin; Vlkolinsky, Roman; Bajo, Michal; Prier, Christopher K; Xiao, Kai-Jiong; Cravatt, Benjamin F; Roberto, Marisa; Baran, Phil S

Stereoretentive radical cross-coupling

立体保持自由基交叉偶联

Sun, Jiawei; He, Jiayan; Massaro, Luca; Cagan, David A; Tsien, Jet; Wang, Yu; Attard, Flynn C; Smith, Jillian E; Lee, Jason S; Kawamata, Yu; Baran, Phil S

Accelerating Medicinal Chemistry: A C(sp(3))-Rich Fragment Toolbox for Redox-Neutral Cross-Coupling

加速药物化学:富含 AC(sp(3)) 的片段工具箱用于氧化还原中性交叉偶联

Tsien, Jet; Péter, Áron; Zeng, Xin; Wang, Shuanghu; Jiang, Baiyang; Emmanuel, Megan A; Oderinde, Martins S; Bolduc, Philippe N; Nicastri, Michael C; Dey, Shalini; Collins, Michael R; Lee, Johnny W; Bravo, Martin; Richardson, Paul F; Sach, Neal W; Bernier, Louise; Palkowitz, Maximilian D; Qiao, Jennifer X; Kawamata, Yu; Baran, Phil S

10-Step, Gram-Scale Total Synthesis of (-)-Bipinnatin J

10步克级(-)-Bipinnatin J全合成

Rodriguez, Anthony J; Pokle, Maithili S; Barnes, Griffin L; Baran, Phil S

Enantiocontrolled Azetidine Library Synthesis via Strain-Release Functionalization of 1-Azabicyclobutanes

通过1-氮杂双环丁烷的应变释放功能化合成对映选择性氮杂环丁烷库

Bielecki, Michael; Nassir, Molhm; Sharma, Hayden A; Truax, Nathanyal J; Raheja, Nicholas; Thompson, Ty M; El-Hayek Ewing, Tamara; Melillo, Bruno; Cravatt, Benjamin F; Baran, Phil S

Pharmacological targeting of RIG-I can selectively activate the integrated stress response

通过药物靶向RIG-I可以选择性地激活整合应激反应。

Cuoco, Caroline A; Ren, Wen; Baron, Kelsey R; Gologo, Sakina; Perea, Valerie; Mathur, Prakhyat; Bora, Prerona; Ta, Amina; Chu, Alan; Aldakhlallah, Rama; Rhoades, Derek; Cole, Christian M; Tan, Ee Phie; Hou, William C; Yoon, Leonard; Guo, Xiaoyan; Rosarda, Jessica D; Baran, Phil S; Kampmann, Martin; Tillery, Lakeisha; Johnson, Kristen A; Powers, Evan T; Wiseman, R Luke; Kelly, Jeffery W

Dibromocarbene addition to bicyclo[1.1.0]butanes: A facile route to substituted bicyclo[1.1.1]pentanes

二溴卡宾与双环[1.1.0]丁烷的加成反应:一种简便合成取代双环[1.1.1]戊烷的方法

Attard, Flynn C; Slobodianyk, Andrii; Bychek, Roman; Panasiuk, Yaroslav; Neigenfind, Philipp; Massaro, Luca; Gardiner, Michael G; Levterov, Vadym V; Baran, Phil S; Mykhailiuk, Pavel K; Malins, Lara R

diAcCA, a Pro-Drug for Carnosic Acid That Activates the Nrf2 Transcriptional Pathway, Shows Efficacy in the 5xFAD Transgenic Mouse Model of Alzheimer's Disease.

diAcCA 是一种激活 Nrf2 转录通路的肌肽酸前药,在 5xFAD 阿尔茨海默病转基因小鼠模型中显示出疗效

Banerjee Piu, Wang Yubo, Carnevale Lauren N, Patel Parth, Raspur Charlene K, Tran Nancy, Zhang Xu, Natarajan Ravi, Roberts Amanda J, Baran Phil S, Lipton Stuart A