日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Artemisinin pressure in field isolates can select highly resistant Plasmodium falciparum parasites with unconventional phenotype and no K13 mutation

在田间分离株中,青蒿素压力可筛选出具有非常规表型且无K13突变的强耐药性恶性疟原虫。

Paloque, Lucie; Mathieu, Luana; Laurent, Marion; Coppée, Romain; Blandin, Stéphanie; Campagne, Pascal; Augereau, Jean-Michel; Musset, Lise; Benoit-Vical, Françoise

Hybrid Molecules as Efficient Drugs against Multidrug-Resistant Malaria Parasites

杂合分子作为对抗多重耐药疟原虫的有效药物

Robert, Anne; Paloque, Lucie; Augereau, Jean-Michel; Nardella, Flore; Nguyen, Michel; Meunier, Bernard; Benoit-Vical, Françoise

Hybrid Peptide-Alkoxyamine Drugs: A Strategy for the Development of a New Family of Antiplasmodial Drugs

肽-烷氧胺杂合药物:开发新型抗疟药物的策略

Embo-Ibouanga, Ange W; Nguyen, Michel; Paloque, Lucie; Coustets, Mathilde; Joly, Jean-Patrick; Augereau, Jean-Michel; Vanthuyne, Nicolas; Bikanga, Raphaël; Coquin, Naomie; Robert, Anne; Audran, Gérard; Boissier, Jérôme; Mellet, Philippe; Benoit-Vical, Françoise; Marque, Sylvain R A

Characterization of antimalarial activity of artemisinin-based hybrid drugs

青蒿素类杂合药物抗疟活性的表征

Quadros, Helenita Costa; Herrmann, Lars; Manaranche, Jeanne; Paloque, Lucie; Borges-Silva, Mariana C; Dziwornu, Godwin Akpeko; D'Alessandro, Sarah; Chibale, Kelly; Basilico, Nicoletta; Benoit-Vical, Françoise; Tsogoeva, Svetlana B; Moreira, Diogo Rodrigo M

In artemisinin-resistant falciparum malaria parasites, mitochondrial metabolic pathways are essential for survival but not those of apicoplast

在对青蒿素产生耐药性的恶性疟原虫中,线粒体代谢途径对其生存至关重要,而顶质体代谢途径则并非如此。

Manel Ouji ,Thibaud Reyser ,Yoshiki Yamaryo-Botté ,Michel Nguyen ,David Rengel ,Axelle Dutreuil ,Marlène Marcellin ,Odile Burlet-Schiltz ,Jean-Michel Augereau ,Michael K Riscoe ,Lucie Paloque ,Cyrille Botté ,Françoise Benoit-Vical

In vitro evaluation of ganaplacide/lumefantrine combination against Plasmodium falciparum in a context of artemisinin resistance

在青蒿素耐药的背景下,对加那普拉西德/卢美芬汀联合用药体外评价其对恶性疟原虫的疗效。

Manaranche, Jeanne; Laurent, Marion; Tressieres, Roxane; Nguyen, Michel; Salim, Maryam; Ouji, Manel; Reyser, Thibaud; Egwu, Chinedu O; Robert, Anne; Augereau, Jean-Michel; Benoit-Vical, Françoise; Paloque, Lucie

Epigenetic regulation as a therapeutic target in the malaria parasite Plasmodium falciparum

表观遗传调控作为疟原虫(恶性疟原虫)的治疗靶点

Reyser, Thibaud; Paloque, Lucie; Augereau, Jean-Michel; Di Stefano, Luisa; Benoit-Vical, Françoise

Epidrugs as Promising Tools to Eliminate Plasmodium falciparum Artemisinin-Resistant and Quiescent Parasites

Epidrugs 是消灭恶性疟原虫青蒿素抗性和休眠寄生虫的有效工具

Thibaud Reyser, Lucie Paloque, Michel Nguyen, Jean-Michel Augereau, Matthew John Fuchter, Marie Lopez, Paola B Arimondo, Storm Hassell-Hart, John Spencer, Luisa Di Stefano, Françoise Benoit-Vical

Mutation in the Plasmodium falciparum BTB/POZ Domain of K13 Protein Confers Artemisinin Resistance

恶性疟原虫K13蛋白BTB/POZ结构域的突变赋予其对青蒿素的耐药性。

Paloque, Lucie; Coppée, Romain; Stokes, Barbara H; Gnädig, Nina F; Niaré, Karamoko; Augereau, Jean-Michel; Fidock, David A; Clain, Jérôme; Benoit-Vical, Françoise

In Vitro and In Silico Antimalarial Evaluation of FM-AZ, a New Artemisinin Derivative

新型青蒿素衍生物 FM-AZ 的体外和计算机模拟抗疟效果评价

Ioannis Tsamesidis, Farnoush Mousavizadeh, Chinedu O Egwu, Dionysia Amanatidou, Antonella Pantaleo, Françoise Benoit-Vical, Karine Reybier, Athanassios Giannis