Novel Autotaxin Inhibitors for the Treatment of Osteoarthritis Pain: Lead Optimization via Structure-Based Drug Design
用于治疗骨关节炎疼痛的新型自泌素抑制剂:基于结构的药物设计优化先导化合物
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.6b00207
Jones, Spencer B; Pfeifer, Lance A; Bleisch, Thomas J; Beauchamp, Thomas J; Durbin, Jim D; Klimkowski, V Joseph; Hughes, Norman E; Rito, Christopher J; Dao, Yen; Gruber, Joseph M; Bui, Hai; Chambers, Mark G; Chandrasekhar, Srinivasan; Lin, Chaohua; McCann, Denis J; Mudra, Daniel R; Oskins, Jennifer L; Swearingen, Craig A; Thirunavukkarasu, Kannan; Norman, Bryan H