日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Consequences of Peptide Macrocyclization Revealed by Virus-Inspired β-Hairpin Mimetics

病毒启发式β-发夹模拟物揭示肽大环化的影响

Bula, Anna L; Bobrovs, Raitis; Arsenyan, Pavel; Pantelejevs, Teodors

Discovery and optimisation of pyrazolo[1,5-a]pyrimidines as aryl hydrocarbon receptor antagonists

发现和优化吡唑并[1,5-a]嘧啶类化合物作为芳烃受体拮抗剂

Bobrovs, Raitis; Terentjeva, Svetlana; Olafsen, Ninni Elise; Dambrauskas, Zilvinas; Gulbinas, Antanas; Maimets, Toivo; Teino, Indrek; Jirgensons, Aigars; Matthews, Jason; Jaudzems, Kristaps

Structural Basis for Inhibition of the SARS-CoV-2 nsp16 by Substrate-Based Dual Site Inhibitors

基于底物的双位点抑制剂抑制SARS-CoV-2 nsp16的结构基础

Kalnins, Gints; Rudusa, Laura; Bula, Anna L; Zelencova-Gopejenko, Diana; Bobileva, Olga; Sisovs, Mihails; Tars, Kaspars; Jirgensons, Aigars; Jaudzems, Kristaps; Bobrovs, Raitis

AlphaFold-SFA: Accelerated sampling of cryptic pocket opening, protein-ligand binding and allostery by AlphaFold, slow feature analysis and metadynamics

AlphaFold-SFA:通过 AlphaFold、慢特征分析和元动力学加速隐蔽口袋开放、蛋白质-配体结合和变构的采样

Vats, Shray; Bobrovs, Raitis; Söderhjelm, Pär; Bhakat, Soumendranath

Structure-based identification of salicylic acid derivatives as malarial threonyl tRNA-synthetase inhibitors.

基于结构的鉴定水杨酸衍生物作为疟疾苏氨酰tRNA合成酶抑制剂

Bobrovs Raitis, Bolsakova Jekaterina, Buitrago Jhon Alexander Rodriguez, Varaceva Larisa, Skvorcova Marija, Kanepe Iveta, Rudnickiha Anastasija, Parisini Emilio, Jirgensons Aigars

Aggregation Condition-Structure Relationship of Mouse Prion Protein Fibrils

小鼠朊病毒蛋白原纤维的聚集条件-结构关系

Fridmanis, Jēkabs; Toleikis, Zigmantas; Sneideris, Tomas; Ziaunys, Mantas; Bobrovs, Raitis; Smirnovas, Vytautas; Jaudzems, Kristaps

Structural and Functional Analysis of BBA03, Borrelia burgdorferi Competitive Advantage Promoting Outer Surface Lipoprotein

伯氏疏螺旋体竞争优势促进蛋白BBA03的结构和功能分析

Fridmanis, Jēkabs; Bobrovs, Raitis; Brangulis, Kalvis; Tārs, Kaspars; Jaudzems, Kristaps