日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In vitro evaluation of the immunogenic potential of gramicidin S and its photocontrolled analogues.

体外评价革兰氏菌素 S 及其光控类似物的免疫原性

Horbatok Kateryna, Semchuk Iryna, Horbach Oleksandr, Khranovska Natalia, Kosach Viktoriia, Borysko Petro, Koniev Serhii, Ulrich Anne S, Afonin Sergii, Komarov Igor V

CF(3)-Cyclobutanes: Synthesis, Properties, and Evaluation as a Unique tert-Butyl Group Analogue

CF(3)-环丁烷:合成、性质及作为独特的叔丁基类似物的评价

Ahunovych, Volodymyr; Klipkov, Anton A; Bugera, Maksym; Tarasenko, Karen; Trofymchuk, Serhii; Razhyk, Bohdan; Boretskyi, Andrii; Stanko, Oleh; Panasiuk, Yaroslav; Shablykin, Oleh; Al-Maali, Galeb; Lesyk, Dmytro; Klymenko-Ulianov, Oleksii; Horbatok, Kateryna; Bodenchuk, Iryna; Kosach, Viktoriia; Borysko, Petro; Kubyshkin, Vladimir; Mykhailiuk, Pavel K

In Vitro Evaluation of In Silico Screening Approaches in Search for Selective ACE2 Binding Chemical Probes

体外评估计算机筛选方法寻找选择性 ACE2 结合化学探针

Alexey V Rayevsky, Andrii S Poturai, Iryna O Kravets, Alexander E Pashenko, Tatiana A Borisova, Ganna M Tolstanova, Dmitriy M Volochnyuk, Petro O Borysko, Olga B Vadzyuk, Diana O Alieksieieva, Yuliana Zabolotna, Olga Klimchuk, Dragos Horvath, Gilles Marcou, Sergey V Ryabukhin, Alexandre Varnek

Further validation of strecker-type α-aminonitriles as a new class of potent human carbonic anhydrase II inhibitors: hit expansion within the public domain using differential scanning fluorimetry leads to chemotype refinement

进一步验证 Strecker 型 α-氨基腈作为一类新型强效人类碳酸酐酶 II 抑制剂的有效性:使用差示扫描荧光法在公共领域内进行匹配扩展可实现化学型细化

Mikhail Krasavin, Stanislav Kalinin, Sergey Zozulya, Anastasia Griniukova, Petro Borysko, Andrea Angeli, Claudiu T Supuran

Screening of benzenesulfonamide in combination with chemically diverse fragments against carbonic anhydrase by differential scanning fluorimetry

用差示扫描荧光法筛选苯磺酰胺与化学性质不同的抗碳酸酐酶片段的组合

Mikhail Krasavin, Stanislav Kalinin, Sergey Zozulya, Anastasiia Gryniukova, Petro Borysko, Andrea Angeli, Claudiu T Supuran

SAR by Space: Enriching Hit Sets from the Chemical Space

空间 SAR:从化学空间丰富命中集

Franca-Maria Klingler, Marcus Gastreich, Oleksandr O Grygorenko, Olena Savych, Petro Borysko, Anastasia Griniukova, Kateryna E Gubina, Christian Lemmen, Yurii S Moroz

Human cytomegalovirus resistance to deoxyribosylindole nucleosides maps to a transversion mutation in the terminase subunit-encoding gene UL89

人类巨细胞病毒对脱氧核糖基吲哚核苷的耐药性定位于末端酶亚基编码基因UL89的颠换突变。

Gentry, Brian G; Phan, Quang; Hall, Ellie D; Breitenbach, Julie M; Borysko, Katherine Z; Kamil, Jeremy P; Townsend, Leroy B; Drach, John C

Resistance of human cytomegalovirus to cyclopropavir maps to a base pair deletion in the open reading frame of UL97

人类巨细胞病毒对环丙沙星的耐药性定位于UL97开放阅读框中的一个碱基对缺失。

Gentry, Brian G; Vollmer, Laura E; Hall, Ellie D; Borysko, Katherine Z; Zemlicka, Jiri; Kamil, Jeremy P; Drach, John C

Synthesis, transport and antiviral activity of Ala-Ser and Val-Ser prodrugs of cidofovir

西多福韦Ala-Ser和Val-Ser前药的合成、转运和抗病毒活性

Peterson, Larryn W; Kim, Jae-Seung; Kijek, Paul; Mitchell, Stefanie; Hilfinger, John; Breitenbach, Julie; Borysko, Kathy; Drach, John C; Kashemirov, Boris A; McKenna, Charles E

Synthesis and biological activation of an ethylene glycol-linked amino acid conjugate of cyclic cidofovir

环状西多福韦乙二醇连接氨基酸缀合物的合成及生物活化

Eriksson, Ulrika; Hilfinger, John M; Kim, Jae-Seung; Mitchell, Stefanie; Kijek, Paul; Borysko, Katherine Z; Breitenbach, Julie M; Drach, John C; Kashemirov, Boris A; McKenna, Charles E