日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Monovalent Lectin Microvirin Utilizes Hydropathic Recognition of HIV-1 Env for Inhibition of Virus Cell Infection

单价凝集素Microvirin利用其对HIV-1 Env的疏水性识别来抑制病毒细胞感染

Bibek Parajuli ,Kriti Acharya ,Harry Charles Bach ,Shiyu Zhang ,Cameron F Abrams ,Irwin Chaiken

Pharmacophore Variants of the Macrocyclic Peptide Triazole Inactivator of HIV-1 Env

HIV-1 包膜蛋白大环肽三唑灭活剂的药效团变体

Monisha Gupta, Gabriela Canziani, Charles Ang, Mohammadjavad Mohammadi, Cameron F Abrams, Derek Yang, Amos B Smith 3rd, Irwin Chaiken

Peptide Triazole Thiol Irreversibly Inactivates Metastable HIV-1 Env by Accessing Conformational Triggers Intrinsic to Virus-Cell Entry

肽三唑硫醇通过进入病毒细胞固有的构象触发因素不可逆地灭活亚稳态 HIV-1 Env

Charles Gotuaco Ang, Erik Carter, Ann Haftl, Shiyu Zhang, Adel A Rashad, Michele Kutzler, Cameron F Abrams, Irwin M Chaiken

Metastable HIV-1 Surface Protein Env Sensitizes Cell Membranes to Transformation and Poration by Dual-Acting Virucidal Entry Inhibitors

亚稳态HIV-1表面蛋白Env使细胞膜对双效杀病毒进入抑制剂的转化和穿孔作用更加敏感

Charles G Ang,Md Alamgir Hossain,Marg Rajpara,Harry Bach,Kriti Acharya,Alexej Dick,Adel A Rashad,Michele Kutzler,Cameron F Abrams,Irwin Chaiken

Restricted HIV-1 Env glycan engagement by lectin-reengineered DAVEI protein chimera is sufficient for lytic inactivation of the virus

经凝集素改造的DAVEI蛋白嵌合体对HIV-1 Env糖基化的特异性结合足以导致病毒裂解性失活。

Bibek Parajuli ,Kriti Acharya ,Harry C Bach ,Bijay Parajuli ,Shiyu Zhang ,Amos B Smith 3rd ,Cameron F Abrams ,Irwin Chaiken

Lytic Inactivation of Human Immunodeficiency Virus by Dual Engagement of gp120 and gp41 Domains in the Virus Env Protein Trimer

病毒包膜蛋白三聚体中gp120和gp41结构域的双重结合导致人类免疫缺陷病毒的裂解性失活

Bibek Parajuli ,Kriti Acharya ,Reina Yu ,Brendon Ngo ,Adel A Rashad ,Cameron F Abrams ,Irwin M Chaiken

Covalent conjugation of a peptide triazole to HIV-1 gp120 enables intramolecular binding site occupancy

肽三唑与 HIV-1 gp120 的共价结合可实现分子内结合位点占据

Ali Emileh, Caitlin Duffy, Andrew P Holmes, Arangassery Rosemary Bastian, Rachna Aneja, Ferit Tuzer, Srivats Rajagopal, Huiyuan Li, Cameron F Abrams, Irwin M Chaiken

A model of peptide triazole entry inhibitor binding to HIV-1 gp120 and the mechanism of bridging sheet disruption

肽三唑进入抑制剂与HIV-1 gp120结合的模型及桥接片破坏机制

Ali Emileh, Ferit Tuzer, Herman Yeh, Muddegowda Umashankara, Diogo R M Moreira, Judith M Lalonde, Carole A Bewley, Cameron F Abrams, Irwin M Chaiken