日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Loss of Integrin-Linked Kinase Sensitizes Breast Cancer to SRC Inhibitors

整合素连接激酶的缺失使乳腺癌对 SRC 抑制剂敏感

Henry Beetham, Billie G C Griffith, Olga Murina, Alexander E P Loftus, David A Parry, Carolin Temps, Jayne Culley, Morwenna Muir, Asier Unciti-Broceta, Andrew H Sims, Adam Byron, Valerie G Brunton

A Conformation Selective Mode of Inhibiting SRC Improves Drug Efficacy and Tolerability

抑制SRC的构象选择性模式可提高药物疗效和耐受性

Carolin Temps, Daniel Lietha, Emily R Webb #, Xue-Feng Li #, John C Dawson #, Morwenna Muir, Kenneth G Macleod, Teresa Valero, Alison F Munro, Rafael Contreras-Montoya, Juan R Luque-Ortega, Craig Fraser, Henry Beetham, Christina Schoenherr, Maria Lopalco, Mark J Arends, Margaret C Frame, Bin-Zhi Qia

An ErbB2/c-Src axis links bioenergetics with PRC2 translation to drive epigenetic reprogramming and mammary tumorigenesis

ErbB2/c-Src 轴将生物能量学与 PRC2 翻译联系起来,以驱动表观遗传重编程和乳腺肿瘤发生

Harvey W Smith, Alison Hirukawa, Virginie Sanguin-Gendreau, Ipshita Nandi, Catherine R Dufour, Dongmei Zuo, Kristofferson Tandoc, Matthew Leibovitch, Salendra Singh, Jonathan P Rennhack, Matthew Swiatnicki, Cynthia Lavoie, Vasilios Papavasiliou, Carolin Temps, Neil O Carragher, Asier Unciti-Broceta,