日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase Inhibition

2-苯基喹啉类化合物通过抑制非结构蛋白13解旋酶发挥抗严重急性呼吸综合征冠状病毒2活性

Cernicchi, Giada; Nizi, Maria Giulia; Emmolo, Roberta; Persoons, Leentje; Laporte, Manon; Jochmans, Dirk; Romeo, Isabella; Pepe, Giacomo; Milite, Ciro; Campiglia, Pietro; Spezzini, Jacopo; Martelli, Alma; Brogi, Simone; Esposito, Francesca; Felicetti, Tommaso; Massari, Serena; Manfroni, Giuseppe; Sabatini, Stefano; Sbardella, Gianluca; Alcaro, Stefano; Neyts, Johan; Corona, Angela; Tramontano, Enzo; De Jonghe, Steven; Tabarrini, Oriana

In Vitro and In Vivo Investigations into the Potential of Quinazoline and Quinoline Derivatives as NorA Efflux Pump Inhibitors Against Resistant Staphylococcus aureus Strains

体外和体内研究喹唑啉及其衍生物作为NorA外排泵抑制剂对抗耐药金黄色葡萄球菌菌株的潜力

Chandal, Nishtha; Sharma, Nidhi; Cernicchi, Giada; Felicetti, Tommaso; Rondini, Tommaso; Acito, Mattia; Nandanwar, Hemraj; Sabatini, Stefano

NorA Efflux Pump Inhibitors: Expanding SAR Knowledge of Pyrazolo[4,3-c][1,2]benzothiazine 5,5-Dioxide Derivatives

NorA 外排泵抑制剂:扩展吡唑并[4,3-c][1,2]苯并噻嗪 5,5-二氧化物衍生物的构效关系知识

Cernicchi, Giada; Di Gregorio, Alessandra; Felicetti, Tommaso; Rampacci, Elisa; Casari, Giulia; Armeni, Tatiana; Romaldi, Brenda; Zefaj, Ermelinda; Passamonti, Fabrizio; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Vignaroli, Carla; Sabatini, Stefano

Inhibition of Staphylococcus pseudintermedius Efflux Pumps by Using Staphylococcus aureus NorA Efflux Pump Inhibitors

利用金黄色葡萄球菌NorA外排泵抑制剂抑制中间葡萄球菌外排泵

Rampacci, Elisa; Felicetti, Tommaso; Cernicchi, Giada; Stefanetti, Valentina; Sabatini, Stefano; Passamonti, Fabrizio