日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of mCMV280: An Oral Ectoparasiticide in the Isoxazoline Class with Reduced Mammalian Brain Exposure

mCMV280 的发现:一种异噁唑啉类口服体外寄生虫杀灭剂,可降低哺乳动物大脑暴露量

McComic, Sarah E; Wilson, Katy B; Li, Zhilin; Chen, Jeffrey; Weiss, Frank; Song, Lirui; Mazumdar, Wrickban; Dvorak, Curt A; Brittain, Jason; Lee, Kyoung-Jin; Li, Shuangwei; Joseph, Sean B; McNamara, Case W; Vos, Martijn W; Sheshachalam, Avinash; Inácio, Alex; Dechering, Koen J; Chatterjee, Arnab K; Swale, Daniel R

NS5-targeting nucleoside analogs inhibit dengue virus and other flaviviruses

靶向NS5的核苷类似物可抑制登革病毒和其他黄病毒

Bhakt, Priyanka; Pokharel, Swechha M; Li, Yue; Srivastava, Tamanna; Miller, Jesse; Dittmar, Mark; Zhu, Yongqing; Nguyen, David; Walter, Zachary; Ayyanathan, Kasirajan; Tudor, Matthew; Yu, Chenguang; Chatterjee, Arnab K; Ramage, Holly; Schultz, David; Cherry, Sara

Minimum inoculum of resistance assay for evaluating for anti-toxoplasmosis compounds that target phenyl alanine tRNA synthetase

用于评估靶向苯丙氨酸tRNA合成酶的抗弓形虫化合物的最低接种量抗性测定

Uddin, Taher; Mittal, Payal; Xie, Han; Melillo, Bruno; Sharma, Amit; Chatterjee, Arnab K; Sibley, L David

SuFEx-based antitubercular compound irreversibly inhibits Pks13

基于 SuFEx 的抗结核化合物不可逆地抑制 Pks13

Krieger, Inna V; Sukheja, Paridhi; Yang, Baiyuan; Tang, Su; Selle, Daniel; Woods, Ashley; Engelhart, Curtis; Kumar, Pradeep; Harbut, Michael B; Liu, Dongdong; Tsuda, Brendan; Qin, Bo; Bare, Grant A L; Li, Gencheng; Chi, Victor; Gambacurta, Julian; Hvizdos, Janine; Reagan, Matthew; Jones, Isabelle L; Massoudi, Lisa M; Woolhiser, Lisa K; Cascioferro, Alessandro; Kundrick, Erica; Singh, Parul; Reiley, William; Ioerger, Thomas R; Kandula, Dilipkumar Reddy; McCabe, Jacob W; Guo, Taijie; Alland, David; Boshoff, Helena I; Schnappinger, Dirk; Robertson, Gregory T; Mdluli, Khisi; Lee, Kyoung-Jin; Dong, Jiajia; Li, Shuangwei; Schultz, Peter G; Joseph, Sean B; Love, Melissa S; Sharpless, K Barry; Petrassi, H Michael; Chatterjee, Arnab K; Sacchettini, James C; McNamara, Case W

Covalent Probes Reveal Small-Molecule Binding Pockets in Structured RNA and Enable Bioactive Compound Design

共价探针揭示结构化RNA中的小分子结合口袋,并实现生物活性化合物的设计

Kovachka, Sandra; Wang, Jielei; Taghavi, Amirhossein; Jia, Yilin; Asaba, Taro; Wolff, Karen C; Martin, Mason; Yang, Xueyi; Meyer, Samantha M; Ottilie, Sabine; Heacock, Mina; Cheng, Zhong; McNamara, Case W; Dubey, Gurudutt; Chatterjee, Arnab K; Chanda, Sumit; Gallego, José; Childs-Disney, Jessica L; Disney, Matthew D

Improved Bicyclic Pyrrolidine Analogues Inhibit Toxoplasma gondii Growth In Vitro and Cure Infection In Vivo

改良的双环吡咯烷类似物在体外抑制弓形虫生长并在体内治愈感染

Uddin, Taher; Xie, Han; Mittal, Payal; Ence, Chloe C; Patil, Shrushti; Sharma, Amit; Melillo, Bruno; Chatterjee, Arnab K; Sibley, L David

A drug repurposing approach reveals targetable epigenetic pathways in Plasmodium vivax hypnozoites.

药物再利用方法揭示了间日疟原虫休眠子中可靶向的表观遗传通路

Maher Steven P, Bakowski Malina A, Vantaux Amélie, Flannery Erika L, Andolina Chiara, Gupta Mohit, Antonova-Koch Yevgeniya, Argomaniz Magdalena, Cabrera-Mora Monica, Campo Brice, Chao Alexander T, Chatterjee Arnab K, Cheng Wayne T, Chuenchob Vorada, Cooper Caitlin A, Cottier Karissa, Galinski Mary R, Harupa-Chung Anke, Ji Hana, Joseph Sean B, Lenz Todd, Lonardi Stefano, Matheson Jessica, Mikolajczak Sebastian A, Moeller Timothy, Orban Agnes, Padín-Irizarry Vivian, Pan Kastin, Péneau Julie, Prudhomme Jacques, Roesch Camille, Ruberto Anthony, Sabnis Saniya S, Saney Celia L, Sattabongkot Jetsumon, Sereshki Saleh, Suriyakan Sangrawee, Ubalee Ratawan, Wang Yinsheng, Wasisakun Praphan, Yin Jiekai, Popovici Jean, McNamara Case W, Joyner Chester, Nosten François H, Witkowski Benoît, Le Roch Karine G, Kyle Dennis E

Design, Synthesis, and Biological Evaluation of Tetrazol-2-yl-acetamides as Novel Antitubercular Agents

四唑-2-基乙酰胺类化合物作为新型抗结核药物的设计、合成及生物学评价

Yang, Baiyuan; Sukheja, Paridhi; Webb, Jasmine; Nguyen-Tran, Van; Chi, Victor; Roszkowski, Emma K; VanderVen, Brian C; Chatterjee, Arnab K; McNamara, Case W

High-Throughput Repurposing Screen Reveals Compounds with Activity against Toxoplasma gondii Bradyzoites.

高通量药物重定位筛选揭示了对弓形虫缓殖子具有活性的化合物

Uddin Taher, Xia Jing, Fu Yong, McNamara Case W, Chatterjee Arnab K, Sibley L David

Bunyaviral Cap-Snatching Endonuclease Activity and Inhibition with Baloxavir-like Inhibitors in the Context of Full-Length L Proteins

在全长L蛋白背景下,布尼亚病毒帽夺取核酸内切酶活性及其与巴洛沙韦样抑制剂的抑制作用

Loutan, Arlo J; Yang, Baiuyan; Connolly, Gabrielle; Montoya, Adam; Smiley, Robert J; Chatterjee, Arnab K; Götte, Matthias