日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Collaborative Virtual Screening Identifies a 2-Aryl-4-aminoquinazoline Series with Efficacy in an In Vivo Model of Trypanosoma cruzi Infection

协同虚拟筛选鉴定出在克氏锥虫感染体内模型中有效的 2-芳基-4-氨基喹唑啉系列

Taisuke Tawaraishi, Atsuko Ochida, Yuichiro Akao, Sachiko Itono, Masahiro Kamaura, Thamina Akther, Mitsuyuki Shimada, Stacie Canan, Sanjoy Chowdhury, Yafeng Cao, Kevin Condroski, Ola Engkvist, Amanda Francisco, Sunil Ghosh, Rina Kaki, John M Kelly, Chiaki Kimura, Thierry Kogej, Kazuya Nagaoka, Akira

Emergence and Targeting of Acquired and Hereditary Resistance to Multikinase RET Inhibition in Patients With RET-Altered Cancer

RET 基因改变癌症患者获得性和遗传性多激酶 RET 抑制剂耐药性的出现及靶向治疗

Wirth, Lori J; Kohno, Takashi; Udagawa, Hibiki; Matsumoto, Shingo; Ishii, Genichiro; Ebata, Kevin; Tuch, Brian B; Zhu, Edward Y; Nguyen, Michele; Smith, Steve; Hanson, Lauren M; Burkard, Michael R; Cable, LouAnn; Blake, James F; Condroski, Kevin R; Brandhuber, Barbara J; Andrews, Steve; Rothenberg, S Michael; Goto, Koichi

Novel Series of Potent Glucokinase Activators Leading to the Discovery of AM-2394

新型强效葡萄糖激酶激活剂系列研究促成了AM-2394的发现

Dransfield, Paul J; Pattaropong, Vatee; Lai, Sujen; Fu, Zice; Kohn, Todd J; Du, Xiaohui; Cheng, Alan; Xiong, Yumei; Komorowski, Renee; Jin, Lixia; Conn, Marion; Tien, Eric; DeWolf, Walter E Jr; Hinklin, Ronald J; Aicher, Thomas D; Kraser, Christopher F; Boyd, Steven A; Voegtli, Walter C; Condroski, Kevin R; Veniant-Ellison, Murielle; Medina, Julio C; Houze, Jonathan; Coward, Peter

C5-Alkyl-2-methylurea-Substituted Pyridines as a New Class of Glucokinase Activators

C5-烷基-2-甲基脲取代的吡啶类化合物作为一类新型葡萄糖激酶激活剂

Du, Xiaohui; Hinklin, Ronald J; Xiong, Yumei; Dransfield, Paul; Park, Jaehyeon; Kohn, Todd J; Pattaropong, Vatee; Lai, SuJen; Fu, Zice; Jiao, Xianyun; Chow, David; Jin, Lixia; Davda, Jasmine; Veniant, Murielle M; Anderson, Deborah A; Baer, Brian R; Bencsik, Josef R; Boyd, Steven A; Chicarelli, Mark Joseph; Mohr, Peter J; Wang, Bin; Condroski, Kevin R; DeWolf, Walter E; Conn, Marion; Tran, Thanhvien; Yang, Jerry; Aicher, Thomas D; Medina, Julio C; Coward, Peter; Houze, Jonathan B