日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Optimization of Pyridone α-Ketoamides as Inhibitors of the SARS-CoV-2 Main Protease

基于结构的吡啶酮α-酮酰胺类化合物作为SARS-CoV-2主蛋白酶抑制剂的优化

Akula, Ravi Kumar; El Kilani, Haifa; Metzen, Alina; Röske, Judith; Zhang, Kaixuan; Göhl, Matthias; Arisetti, Nanaji; Marsh, Graham P; Maple, Hannah J; Cooper, Mark S; Karadogan, Burhan; Jochmans, Dirk; Neyts, Johan; Rox, Katharina; Hilgenfeld, Rolf; Brönstrup, Mark

Development of p300-targeting degraders with enhanced selectivity and onset of degradation.

开发具有增强选择性和更快降解速度的p300靶向降解剂

Marsh Graham P, Cooper Mark S, Goggins Sean, Reynolds Stephen J, Wheeler Dean F, Cresser-Brown Joel O, Arnold Robert E, Babcock Emily G, Hughes Gareth, Bosnakovski Darko, Kyba Michael, Ojeda Samuel, Harrison Drew A, Ott Christopher J, Maple Hannah J

Skin 11β-hydroxysteroid dehydrogenase type 1 enzyme expression regulates burn wound healing and can be targeted to modify scar characteristics

皮肤11β-羟类固醇脱氢酶1型酶的表达调控烧伤创面愈合,可作为改善瘢痕特征的靶点。

Tsai, Kevin H-Y; Shi, Huaikai; Parungao, Roxanne J; Naficy, Sina; Ding, Xiaotong; Ding, Xiaofeng; Hew, Jonathan J; Wang, Xiaosuo; Chrzanowski, Wojciech; Lavery, Gareth G; Li, Zhe; Issler-Fisher, Andrea C; Chen, Jun; Tan, Qian; Maitz, Peter K; Cooper, Mark S; Wang, Yiwei

Effect of AZD4017, a Selective 11β-HSD1 Inhibitor, on Bone Turnover Markers in Postmenopausal Osteopenia

选择性11β-HSD1抑制剂AZD4017对绝经后骨质减少症患者骨转换标志物的影响

Abbas, Afroze; Schini, Marian; Ainsworth, Gemma; Brown, Sarah R; Oughton, Jamie; Crowley, Rachel K; Cooper, Mark S; Fairclough, Rebecca J; Eastell, Richard; Stewart, Paul M

The contradictory role of androgens in cutaneous and major burn wound healing

雄激素在皮肤和严重烧伤创面愈合中的矛盾作用

Shi, Huaikai; Cheer, Kenny; Simanainen, Ulla; Lesmana, Brian; Ma, Duncan; Hew, Jonathan J; Parungao, Roxanne J; Li, Zhe; Cooper, Mark S; Handelsman, David J; Maitz, Peter K; Wang, Yiwei

Endogenous Glucocorticoid Metabolism in Bone: Friend or Foe

骨骼内源性糖皮质激素代谢:是敌是友

Martin, Claire S; Cooper, Mark S; Hardy, Rowan S

Role of 11β-HSD type 1 in abnormal HPA axis activity during immune-mediated arthritis

11β-HSD 1 型在免疫介导性关节炎中异常 HPA 轴活动中的作用

Sattler, Janko; Tu, Jinwen; Stoner, Shihani; Li, Jingbao; Buttgereit, Frank; Seibel, Markus J; Zhou, Hong; Cooper, Mark S

A Humoral Immune Response Alters the Distribution of Enzyme Replacement Therapy in Murine Mucopolysaccharidosis Type I

体液免疫反应改变小鼠 I 型粘多糖贮积症中酶替代疗法的分布

Steven Q Le, Shih-Hsin Kan, Don Clarke, Valentina Sanghez, Martin Egeland, Kristen N Vondrak, Terence M Doherty, Moin U Vera, Michelina Iacovino, Jonathan D Cooper, Mark S Sands, Patricia I Dickson

Vitamin D deficiency contributes directly to the acute respiratory distress syndrome (ARDS)

维生素D缺乏症直接导致急性呼吸窘迫综合征(ARDS)。

Dancer, Rachel C A; Parekh, Dhruv; Lax, Sian; D'Souza, Vijay; Zheng, Shengxing; Bassford, Chris R; Park, Daniel; Bartis, D G; Mahida, Rahul; Turner, Alice M; Sapey, Elizabeth; Wei, Wenbin; Naidu, Babu; Stewart, Paul M; Fraser, William D; Christopher, Kenneth B; Cooper, Mark S; Gao, Fang; Sansom, David M; Martineau, Adrian R; Perkins, Gavin D; Thickett, David R

Differential glucocorticoid metabolism in patients with persistent versus resolving inflammatory arthritis

持续性炎症性关节炎患者与缓解期炎症性关节炎患者的糖皮质激素代谢差异

Nanus, Dominika E; Filer, Andrew D; Yeo, Lorraine; Scheel-Toellner, Dagmar; Hardy, Rowan; Lavery, Gareth G; Stewart, Paul M; Buckley, Christopher D; Tomlinson, Jeremy W; Cooper, Mark S; Raza, Karim