日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase Inhibition

2-苯基喹啉类化合物通过抑制非结构蛋白13解旋酶发挥抗严重急性呼吸综合征冠状病毒2活性

Cernicchi, Giada; Nizi, Maria Giulia; Emmolo, Roberta; Persoons, Leentje; Laporte, Manon; Jochmans, Dirk; Romeo, Isabella; Pepe, Giacomo; Milite, Ciro; Campiglia, Pietro; Spezzini, Jacopo; Martelli, Alma; Brogi, Simone; Esposito, Francesca; Felicetti, Tommaso; Massari, Serena; Manfroni, Giuseppe; Sabatini, Stefano; Sbardella, Gianluca; Alcaro, Stefano; Neyts, Johan; Corona, Angela; Tramontano, Enzo; De Jonghe, Steven; Tabarrini, Oriana

N-alkyl and N-benzyl indoles are anti-SARS-CoV-2 agents and nsp13 inhibitors

N-烷基和N-苄基吲哚是抗SARS-CoV-2药物和nsp13抑制剂

Albano, Aurora; Emmolo, Roberta; De Santis, Riccardo; Patacchini, Elisa; Madia, Valentina Noemi; Maloccu, Stefania; Ialongo, Davide; Ruggieri, Giuseppe; Arpacioglu, Merve; Scipione, Luigi; Saccoliti, Francesco; Amatore, Donatella; Grilli, Giorgia; Lista, Florigio; Esposito, Francesca; Tramontano, Enzo; Corona, Angela; Di Santo, Roberto; Costi, Roberta

Synthesis and Evaluation of Thiazolidinone-Isatin Hybrids for Selective Inhibition of Cancer-Related Carbonic Anhydrases

噻唑烷酮-靛红杂合物的合成与评价及其对癌症相关碳酸酐酶的选择性抑制作用

Onali, Alessia; Sanna, Erica; Lupia, Antonio; Secci, Daniela; Atzeni, Giulia; Demuru, Laura; Angeli, Andrea; Cottiglia, Filippo; Meleddu, Rita; Emmolo, Roberta; Corona, Angela; Maccioni, Elias; Supuran, Claudiu T; Distinto, Simona

Dual-Site Inhibition of SARS-CoV-2 RNA-Dependent RNA Polymerase by Small Molecules Able to Block Viral Replication Identified through a Computer-Aided Drug Discovery Approach

通过计算机辅助药物发现方法鉴定出能够阻断SARS-CoV-2 RNA依赖性RNA聚合酶双位点抑制的小分子

Malune, Paolo; Iaconis, Daniela; Manelfi, Candida; Giunta, Stefano; Emmolo, Roberta; Lunghini, Filippo; Paulis, Annalaura; Talarico, Carmine; Corona, Angela; Beccari, Andrea Rosario; Tramontano, Enzo; Esposito, Francesca

Thiol-Reactive or Redox-Active: Revising a Repurposing Screen Led to a New Invalidation Pipeline and Identified a True Noncovalent Inhibitor Against Papain-like Protease from SARS-CoV-2.

硫醇反应性或氧化还原活性:修改重新定位筛选导致新的无效化流程,并鉴定出针对 SARS-CoV-2 木瓜蛋白酶样蛋白酶的真正非共价抑制剂

Kuzikov Maria, Morasso Stefano, Reinshagen Jeanette, Wolf Markus, Monaco Vittoria, Cozzolino Flora, Golič Grdadolnik Simona, Šket Primož, Plavec Janez, Iaconis Daniela, Summa Vincenzo, Corona Angela, Paulis Annalaura, Esposito Francesca, Tramontano Enzo, Monti Maria, Beccari Andrea R, Manelfi Candida, Windshügel Björn, Gribbon Philip, Storici Paola, Zaliani Andrea

Structure-Activity Relationships of New 1-Aryl-1H-Indole Derivatives as SARS-CoV-2 Nsp13 Inhibitors

新型1-芳基-1H-吲哚衍生物作为SARS-CoV-2 Nsp13抑制剂的构效关系

Madia, Valentina Noemi; Emmolo, Roberta; Patacchini, Elisa; Amatore, Donatella; Maloccu, Stefania; Ialongo, Davide; Albano, Aurora; Ruggieri, Giuseppe; Cara, Emanuele; Zarbo, Laura; Messore, Antonella; De Santis, Riccardo; Amoroso, Alessandra; Lista, Florigio; Esposito, Francesca; Tramontano, Enzo; Corona, Angela; Di Santo, Roberto; Costi, Roberta

New Thiazolidine-4-One Derivatives as SARS-CoV-2 Main Protease Inhibitors

新型噻唑烷-4-酮衍生物作为SARS-CoV-2主蛋白酶抑制剂

Messore, Antonella; Malune, Paolo; Patacchini, Elisa; Madia, Valentina Noemi; Ialongo, Davide; Arpacioglu, Merve; Albano, Aurora; Ruggieri, Giuseppe; Saccoliti, Francesco; Scipione, Luigi; Tramontano, Enzo; Canton, Serena; Corona, Angela; Scognamiglio, Sante; Paulis, Annalaura; Suleiman, Mustapha; Al-Maqtari, Helmi Mohammed; Abid, Fatma Mohamed A; Kawsar, Sarkar M A; Sankaranarayanan, Murugesan; Di Santo, Roberto; Esposito, Francesca; Costi, Roberta

Structure-Based Design of Novel Thiazolone[3,2-a]pyrimidine Derivatives as Potent RNase H Inhibitors for HIV Therapy

基于结构的噻唑啉酮[3,2-a]嘧啶衍生物新型高效RNase H抑制剂在HIV治疗中的应用

Zhu, Xuan-De; Corona, Angela; Maloccu, Stefania; Tramontano, Enzo; Wang, Shuai; Pannecouque, Christophe; De Clercq, Erik; Meng, Ge; Chen, Fen-Er

Visible Light-Mediated Inactivation of H1N1 Virus UsingPolymer-Based Heterojunction Photocatalyst

利用聚合物基异质结光催化剂实现可见光介导的H1N1病毒灭活

Porcu, Stefania; Maloccu, Stefania; Corona, Angela; Hazra, Moulika; David, Tullia Carla; Chiriu, Daniele; Carbonaro, Carlo Maria; Tramontano, Enzo; Ricci, Pier Carlo

HIV-1 Integrase Inhibition Activity by Spiroketals Derived from Plagius flosculosus, an Endemic Plant of Sardinia (Italy) and Corsica (France)

从意大利撒丁岛和法国科西嘉岛特有植物 Plagius flosculosus 中提取的螺缩酮对 HIV-1 整合酶的抑制活性

Sanna, Cinzia; D'Abrosca, Brigida; Fiorentino, Antonio; Giammarino, Federica; Vicenti, Ilaria; Corona, Angela; Caredda, Alessia; Tramontano, Enzo; Esposito, Francesca