日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Nature-Inspired 1-Phenylpyrrolo[2,1- a]isoquinoline Scaffold for Novel Antiproliferative Agents Circumventing P-Glycoprotein-Dependent Multidrug Resistance

受自然启发的 1-苯基吡咯并[2,1- a]异喹啉支架可用于新型抗增殖药物,以规避 P-糖蛋白依赖性多药耐药性

Alisa A Nevskaya, Rosa Purgatorio, Tatiana N Borisova, Alexey V Varlamov, Lada V Anikina, Arina Yu Obydennik, Elena Yu Nevskaya, Mauro Niso, Nicola A Colabufo, Antonio Carrieri, Marco Catto, Modesto de Candia, Leonid G Voskressensky, Cosimo D Altomare

Synthesis of Novel Benzo[ b][1,6]naphthyridine Derivatives and Investigation of Their Potential as Scaffolds of MAO Inhibitors

新型苯并[b][1,6]萘啶衍生物的合成及其作为 MAO 抑制剂骨架的潜力研究

Larisa N Kulikova, Ghulam Reza Raesi, Daria D Levickaya, Rosa Purgatorio, Gabriella La Spada, Marco Catto, Cosimo D Altomare, Leonid G Voskressensky

Chemical and Biological Evaluation of Novel 1 H-Chromeno[3,2- c]pyridine Derivatives as MAO Inhibitors Endowed with Potential Anticancer Activity

新型 1 H-色烯并[3,2- c]吡啶衍生物作为具有潜在抗癌活性的 MAO 抑制剂的化学和生物学评价

Larisa N Kulikova, Rosa Purgatorio, Andrey A Beloglazkin, Viktor A Tafeenko, Raesi Gh Reza, Daria D Levickaya, Sabina Sblano, Angelina Boccarelli, Modesto de Candia, Marco Catto, Leonid G Voskressensky, Cosimo D Altomare

Synthesis of Isomeric 3-Benzazecines Decorated with Endocyclic Allene Moiety and Exocyclic Conjugated Double Bond and Evaluation of Their Anticholinesterase Activity

环内丙二烯部分和环外共轭双键修饰的异构体3-苯并氮杂环丙烷的合成及其抗胆碱酯酶活性评价

Alexander A Titov, Rosa Purgatorio, Arina Y Obydennik, Anna V Listratova, Tatiana N Borisova, Modesto de Candia, Marco Catto, Cosimo D Altomare, Alexey V Varlamov, Leonid G Voskressensky

Assessing the Role of a Malonamide Linker in the Design of Potent Dual Inhibitors of Factor Xa and Cholinesterases

评估丙二酰胺连接子在设计 Xa 因子和胆碱酯酶强效双重抑制剂中的作用

Rosa Purgatorio, Nicola Gambacorta, Francesco Samarelli, Gianfranco Lopopolo, Modesto de Candia, Marco Catto, Orazio Nicolotti, Cosimo D Altomare

Design, synthesis and biological evaluation of light-driven on-off multitarget AChE and MAO-B inhibitors

光驱动开关多靶点 AChE 和 MAO-B 抑制剂的设计、合成及生物学评价

Marco Paolino, Mariagrazia Rullo, Samuele Maramai, Modesto de Candia, Leonardo Pisani, Marco Catto, Claudia Mugnaini, Antonella Brizzi, Andrea Cappelli, Massimo Olivucci, Federico Corelli, Cosimo D Altomare

Homobivalent Lamellarin-Like Schiff Bases: In Vitro Evaluation of Their Cancer Cell Cytotoxicity and Multitargeting Anti-Alzheimer's Disease Potential

同型二价层状蛋白样席夫碱:体外评估其癌细胞毒性和多靶点抗阿尔茨海默病潜力

Alisa A Nevskaya, Lada V Anikina, Rosa Purgatorio, Marco Catto, Orazio Nicolotti, Modesto de Candia, Leonardo Pisani, Tatiana N Borisova, Almira R Miftyakhova, Aleksey V Varlamov, Elena Yu Nevskaya, Roman S Borisov, Leonid G Voskressensky, Cosimo D Altomare

Synthesis and Biological Evaluation of Dantrolene-Like Hydrazide and Hydrazone Analogues as Multitarget Agents for Neurodegenerative Diseases

丹曲林类酰肼和酰腙类似物的合成及作为神经退行性疾病多靶点药物的生物学评价

Isabella Bolognino, Nicola Giangregorio, Annamaria Tonazzi, Antón L Martínez, Cosimo D Altomare, María I Loza, Sara Sablone, Saverio Cellamare, Marco Catto

Pharmacophore Modeling and 3D-QSAR Study of Indole and Isatin Derivatives as Antiamyloidogenic Agents Targeting Alzheimer's Disease

吲哚和靛蓝衍生物作为抗淀粉样变性药物治疗阿尔茨海默病的药效团建模和 3D-QSAR 研究

Rosa Purgatorio, Nicola Gambacorta, Marco Catto, Modesto de Candia, Leonardo Pisani, Alba Espargaró, Raimon Sabaté, Saverio Cellamare, Orazio Nicolotti, Cosimo D Altomare