日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Short-course combination treatment for experimental chronic Chagas disease

针对实验性慢性恰加斯病的短期联合治疗

González, Silvia; Wall, Richard J; Thomas, John; Braillard, Stephanie; Brunori, Gino; Camino Díaz, Isabel; Cantizani, Juan; Carvalho, Sandra; Castañeda Casado, Pablo; Chatelain, Eric; Cotillo, Ignacio; Fiandor, Jose M; Francisco, Amanda Fortes; Grimsditch, David; Keenan, Martine; Kelly, John M; Kessler, Albane; Luise, Chiara; Lyon, Jon J; MacLean, Lorna; Marco, Maria; Martin, J Julio; Martinez Martinez, Maria S; Paterson, Christy; Read, Kevin D; Santos-Villarejo, Angel; Zuccotto, Fabio; Wyllie, Susan; Miles, Tim J; De Rycker, Manu

Discovery of pyrazolopyrrolidinones as potent, broad-spectrum inhibitors of Leishmania infection

发现吡唑并吡咯烷酮是利什曼原虫感染的强效广谱抑制剂

John A Kavouris, Laura-Isobel McCall, Miriam A Giardini, Geraldine De Muylder, Diane Thomas, Adolfo Garcia-Pérez, Juan Cantizani, Ignacio Cotillo, Jose M Fiandor, James H McKerrow, Camila I De Oliveira, Jair L Siqueira-Neto, Silvia González, Lauren E Brown, Scott E Schaus

Identification and development of a series of disubstituted piperazines for the treatment of Chagas disease

鉴定和开发一系列二取代哌嗪类化合物用于治疗恰加斯病

McGonagle, Kate; Tarver, Gary J; Cantizani, Juan; Cotillo, Ignacio; Dodd, Peter G; Ferguson, Liam; Gilbert, Ian H; Marco, Maria; Miles, Tim; Naylor, Claire; Osuna-Cabello, Maria; Paterson, Christy; Read, Kevin D; Pinto, Erika G; Riley, Jennifer; Scullion, Paul; Shishikura, Yoko; Simeons, Frederick; Stojanovski, Laste; Svensen, Nina; Thomas, John; Wyatt, Paul G; Manzano, Pilar; De Rycker, Manu; Thomas, Michael G

Rate-of-Kill (RoK) assays to triage large compound sets for Chagas disease drug discovery: Application to GSK Chagas Box

利用杀伤率 (RoK) 检测方法筛选用于恰加斯病药物研发的大量化合物:以葛兰素史克恰加斯病盒为例

Cantizani, Juan; Gamallo, Pablo; Cotillo, Ignacio; Alvarez-Velilla, Raquel; Martin, Julio

Development of Trypanosoma cruzi in vitro assays to identify compounds suitable for progression in Chagas' disease drug discovery

开发克氏锥虫体外检测方法,以筛选适合推进恰加斯病药物研发的化合物

MacLean, Lorna M; Thomas, John; Lewis, Michael D; Cotillo, Ignacio; Gray, David W; De Rycker, Manu

2,4-Diamino-6-methylpyrimidines for the potential treatment of Chagas' disease

2,4-二氨基-6-甲基嘧啶类化合物有望用于治疗恰加斯病

Thomas, Michael G; De Rycker, Manu; Cotillo Torrejon, Ignacio; Thomas, John; Riley, Jennifer; Spinks, Daniel; Read, Kevin D; Miles, Tim J; Gilbert, Ian H; Wyatt, Paul G

New compound sets identified from high throughput phenotypic screening against three kinetoplastid parasites: an open resource

通过针对三种动质体寄生虫的高通量表型筛选鉴定出的新化合物集:一种开放资源

Imanol Peña, M Pilar Manzano, Juan Cantizani, Albane Kessler, Julio Alonso-Padilla, Ana I Bardera, Emilio Alvarez, Gonzalo Colmenarejo, Ignacio Cotillo, Irene Roquero, Francisco de Dios-Anton, Vanessa Barroso, Ana Rodriguez, David W Gray, Miguel Navarro, Vinod Kumar, Alexander Sherstnev, David H Dre

Automated high-content assay for compounds selectively toxic to Trypanosoma cruzi in a myoblastic cell line

对成肌细胞系中克氏锥虫具有选择性毒性的化合物进行自动高内涵测定

Julio Alonso-Padilla, Ignacio Cotillo, Jesús L Presa, Juan Cantizani, Imanol Peña, Ana I Bardera, Jose J Martín, Ana Rodriguez