日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Carboxylic Acid Bioisosteres Boost Nurr1 Agonist Selectivity

羧酸生物等排体增强 Nurr1 激动剂选择性

Stiller, Tanja; Gege, Christian; Saeb, Wael; Vietor, Jan; López-García, Úrsula; Busch, Romy; Kohlhof, Hella; Vitt, Daniel; Merk, Daniel

Chemogenomics for steroid hormone receptors (NR3)

类固醇激素受体(NR3)化学基因组学

Espen Schallmayer, Laura Isigkeit, Lewis Elson, Susanne Müller, Stefan Knapp, Julian A Marschner, Daniel Merk

Prospective de novo drug design with deep interactome learning

利用深度相互作用组学习进行前瞻性从头药物设计

Kenneth Atz, Leandro Cotos, Clemens Isert, Maria Håkansson, Dorota Focht, Mattis Hilleke, David F Nippa, Michael Iff, Jann Ledergerber, Carl C G Schiebroek, Valentina Romeo, Jan A Hiss, Daniel Merk, Petra Schneider, Bernd Kuhn, Uwe Grether, Gisbert Schneider

Automated design of multi-target ligands by generative deep learning

通过生成深度学习自动设计多靶点配体

Laura Isigkeit, Tim Hörmann, Espen Schallmayer, Katharina Scholz, Felix F Lillich, Johanna H M Ehrler, Benedikt Hufnagel, Jasmin Büchner, Julian A Marschner, Jörg Pabel, Ewgenij Proschak, Daniel Merk

Chemogenomics for NR1 nuclear hormone receptors

NR1 核激素受体化学基因组学

Laura Isigkeit #, Espen Schallmayer #, Romy Busch, Lorene Brunello, Amelie Menge, Lewis Elson, Susanne Müller, Stefan Knapp, Alexandra Stolz, Julian A Marschner, Daniel Merk

Development of Nurr1 agonists from amodiaquine by scaffold hopping and fragment growing

通过骨架跳跃和片段生长从阿莫地喹开发 Nurr1 激动剂

Minh Sai, Emily C Hank, Hin-Man Tai, Till Kasch, Max Lewandowski, Michelle Vincendeau, Julian A Marschner, Daniel Merk

Dual soluble epoxide hydrolase inhibitor - farnesoid X receptor agonist interventional treatment attenuates renal inflammation and fibrosis

双可溶性环氧化物水解酶抑制剂-法呢醇X受体激动剂介入治疗减轻肾脏炎症和纤维化

Md Abdul Hye Khan, Benjamin Nolan, Anna Stavniichuk, Daniel Merk, John D Imig

De Novo Design of Nurr1 Agonists via Fragment-Augmented Generative Deep Learning in Low-Data Regime

在低数据环境下通过片段增强生成深度学习进行 Nurr1 激动剂的从头设计

Marco Ballarotto, Sabine Willems, Tanja Stiller, Felix Nawa, Julian A Marschner, Francesca Grisoni, Daniel Merk

Development of a Potent Nurr1 Agonist Tool for In Vivo Applications

开发用于体内应用的强效 Nurr1 激动剂工具

Jan Vietor, Christian Gege, Tanja Stiller, Romy Busch, Espen Schallmayer, Hella Kohlhof, Georg Höfner, Jörg Pabel, Julian A Marschner, Daniel Merk

Exploring Fatty Acid Mimetics as NR4A Ligands

探索脂肪酸类似物作为 NR4A 配体

Tanja Stiller, Daniel Merk