日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, and Characterization of New δ Opioid Receptor-Selective Fluorescent Probes and Applications in Single-Molecule Microscopy of Wild-Type Receptors

新型δ阿片受体选择性荧光探针的设计、合成和表征及其在野生型受体单分子显微镜中的应用

Antonios Drakopoulos, Zsombor Koszegi, Kerstin Seier, Harald Hübner, Damien Maurel, Rémy Sounier, Sébastien Granier, Peter Gmeiner, Davide Calebiro, Michael Decker

Plasma membrane preassociation drives β-arrestin coupling to receptors and activation

质膜预结合驱动β-arrestin与受体偶联并活化

Jak Grimes, Zsombor Koszegi, Yann Lanoiselée, Tamara Miljus, Shannon L O'Brien, Tomasz M Stepniewski, Brian Medel-Lacruz, Mithu Baidya, Maria Makarova, Ravi Mistry, Joëlle Goulding, Julia Drube, Carsten Hoffmann, Dylan M Owen, Arun K Shukla, Jana Selent, Stephen J Hill, Davide Calebiro

Revealing the tissue-level complexity of endogenous glucagon-like peptide-1 receptor expression and signaling

揭示内源性胰高血糖素样肽-1受体表达和信号传导的组织水平复杂性

Julia Ast, Daniela Nasteska, Nicholas H F Fine, Daniel J Nieves, Zsombor Koszegi, Yann Lanoiselée, Federica Cuozzo, Katrina Viloria, Andrea Bacon, Nguyet T Luu, Philip N Newsome, Davide Calebiro, Dylan M Owen, Johannes Broichhagen, David J Hodson

Filamin A organizes γ‑aminobutyric acid type B receptors at the plasma membrane

细丝蛋白 A 在质膜上组织 γ-氨基丁酸 B 型受体

Marie-Lise Jobin, Sana Siddig, Zsombor Koszegi, Yann Lanoiselée, Vladimir Khayenko, Titiwat Sungkaworn, Christian Werner, Kerstin Seier, Christin Misigaiski, Giovanna Mantovani, Markus Sauer, Hans M Maric, Davide Calebiro

TSH Pulses Finely Tune Thyroid Hormone Release and TSH Receptor Transduction

TSH 脉冲精细调节甲状腺激素释放和 TSH 受体转导

Anne Guillou, Yasmine Kemkem, Chrystel Lafont, Pierre Fontanaud, Davide Calebiro, Pauline Campos, Xavier Bonnefont, Tatiana Fiordelisio-Coll, Ying Wang, Emilie Brûlé, Daniel J Bernard, Paul Le Tissier, Frederik Steyn, Patrice Mollard

Dimerization of GPCRs: Novel insight into the role of FLNA and SSAs regulating SST2 and SST5 homo- and hetero-dimer formation

GPCR 的二聚化:对 FLNA 和 SSA 调节 SST2 和 SST5 同源二聚体和异源二聚体形成作用的新见解

Donatella Treppiedi, Giusy Marra, Genesio Di Muro, Rosa Catalano, Federica Mangili, Emanuela Esposito, Davide Calebiro, Maura Arosio, Erika Peverelli, Giovanna Mantovani

Lipolysis drives expression of the constitutively active receptor GPR3 to induce adipose thermogenesis

脂肪分解驱动组成型活性受体GPR3的表达,从而诱导脂肪组织产热。

Olivia Sveidahl Johansen ,Tao Ma ,Jakob Bondo Hansen ,Lasse Kruse Markussen ,Renate Schreiber ,Laia Reverte-Salisa ,Hua Dong ,Dan Ploug Christensen ,Wenfei Sun ,Thorsten Gnad ,Iuliia Karavaeva ,Thomas Svava Nielsen ,Sander Kooijman ,Cheryl Cero ,Oksana Dmytriyeva ,Yachen Shen ,Maria Razzoli ,Shannon L O'Brien ,Eline N Kuipers ,Carsten Haagen Nielsen ,William Orchard ,Nienke Willemsen ,Naja Zenius Jespersen ,Morten Lundh ,Elahu Gosney Sustarsic ,Cecilie Mørch Hallgren ,Mikkel Frost ,Seth McGonigle ,Marie Sophie Isidor ,Christa Broholm ,Oluf Pedersen ,Jacob Bo Hansen ,Niels Grarup ,Torben Hansen ,Andreas Kjær ,James G Granneman ,M Madan Babu ,Davide Calebiro ,Søren Nielsen ,Mikael Rydén ,Raymond Soccio ,Patrick C N Rensen ,Jonas Thue Treebak ,Thue Walter Schwartz ,Brice Emanuelli ,Alessandro Bartolomucci ,Alexander Pfeifer ,Rudolf Zechner ,Camilla Scheele ,Susanne Mandrup ,Zachary Gerhart-Hines

PKA Cα subunit mutation triggers caspase-dependent RIIβ subunit degradation via Ser114 phosphorylation

PKA Cα 亚基突变通过 Ser114 磷酸化引发 caspase 依赖的 RIIβ 亚基降解

Isabel Weigand, Cristina L Ronchi, Jens T Vanselow, Kerstin Bathon, Kerstin Lenz, Sabine Herterich, Andreas Schlosser, Matthias Kroiss, Martin Fassnacht, Davide Calebiro, Silviu Sbiera

Spatiotemporal GLP-1 and GIP receptor signaling and trafficking/recycling dynamics induced by selected receptor mono- and dual-agonists

选定受体单和双激动剂诱导的时空 GLP-1 和 GIP 受体信号传导和运输/循环动力学

Aaron Novikoff, Shannon L O'Brien, Miriam Bernecker, Gerald Grandl, Maximilian Kleinert, Patrick J Knerr, Kerstin Stemmer, Martin Klingenspor, Anja Zeigerer, Richard DiMarchi, Matthias H Tschöp, Brian Finan, Davide Calebiro, Timo D Müller

Genomic and sequence variants of protein kinase A regulatory subunit type 1β (PRKAR1B) in patients with adrenocortical disease and Cushing syndrome

肾上腺皮质疾病和库欣综合征患者的蛋白激酶 A 调节亚基 1β 型 (PRKAR1B) 的基因组和序列变异

Ludivine Drougat #, Nikolaos Settas #, Cristina L Ronchi, Kerstin Bathon, Davide Calebiro, Andrea Gutierrez Maria, Sara Haydar, Antonios Voutetakis, Edra London, Fabio R Faucz, Constantine A Stratakis