日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Data-Driven Design of PROTAC Linkers to Improve PROTAC Cell Membrane Permeability.

基于数据驱动的 PROTAC 连接子设计,以提高 PROTAC 细胞膜渗透性。

Murakami Yuki, Ishida Shoichi, Cho Nobuo, Yuki Hitomi, Ohta Masateru, Honma Teruki, Demizu Yosuke, Terayama Kei

Stereochemical and Structural Characterization of Methionine Oxidation in the IgG1 Fc Region by Integrated NMR and LC-MS Analysis

利用核磁共振和液相色谱-质谱联用技术对IgG1 Fc区甲硫氨酸氧化进行立体化学和结构表征

Yagi-Utsumi, Maho; Yanaka, Saeko; Hashii, Noritaka; Tomita, Kohei; Misawa, Takashi; Demizu, Yosuke; Ishii-Watabe, Akiko; Kato, Koichi

Application of HIV-1 viral protein R-derived-peptides as new E3 ligase-binding components of BRD4 degraders

HIV-1病毒蛋白R衍生肽作为BRD4降解剂的新型E3连接酶结合组分的应用

Tsuji, Kohei; Huang, Xueyuan; Miyamoto, Maho; Sukegawa, Sayaka; Yokoo, Hidetomo; Takeuchi, Hiroaki; Demizu, Yosuke; Tamamura, Hirokazu

Shifting Antimicrobial Susceptibility Patterns of Uropathogens: A 20-Year Analysis of Urine Cultures

泌尿道病原体抗菌药物敏感性模式的变化:一项为期20年的尿培养分析

Takebe, Shinichi; Endo, Masami; Demizu, Nanaho; Tokumoto, Mei; Morinaga, Ryota; Mitome, Taku; Takizawa, Akitoshi

Correction: Strategic design of GalNAc-helical peptide ligands for efficient liver targeting

更正:GalNAc螺旋肽配体的策略性设计及其在肝脏靶向治疗中的应用

Ito, Takahito; Ohoka, Nobumichi; Aoyama, Michihiko; Nishikaze, Takashi; Misawa, Takashi; Inoue, Takao; Ishii-Watabe, Akiko; Demizu, Yosuke

High-Resolution HPLC for Separating Peptide-Oligonucleotide Conjugates

高分辨率高效液相色谱法分离肽-寡核苷酸缀合物

Naganuma, Miyako; Tsuji, Genichiro; Amiya, Misato; Hirai, Reira; Higuchi, Yuki; Hata, Naoko; Nozawa, Saoko; Watanabe, Daishi; Nakajima, Taeko; Demizu, Yosuke

Clozapine as an E3 Ligand for PROTAC Technology

氯氮平作为 PROTAC 技术的 E3 配体

Takano, Reina; Ohoka, Nobumichi; Kurohara, Takashi; Arakawa, Noriaki; Ohgane, Kenji; Inoue, Takao; Yokoo, Hidetomo; Demizu, Yosuke

Advances in the development of Wnt/β-catenin signaling inhibitors

Wnt/β-catenin信号通路抑制剂研发进展

Fujita, Minami; Demizu, Yosuke

Optimizing linker rigidity to improve intracellular behavior of PROTACs targeting hematopoietic prostaglandin D synthase.

优化连接子刚性以改善靶向造血前列腺素 D 合成酶的 PROTAC 的细胞内行为

Osawa Hinata, Saito Kosuke, Demizu Yosuke

Combination Treatment with Spacer Placement Surgery Followed by Particle Radiotherapy for Lymph Node Metastasis from Uterine Cancer

子宫癌淋巴结转移的联合治疗:间隔植入手术联合粒子放射治疗

Komatsu, Shohei; Nagamata, Satoshi; Terashima, Kazuki; Demizu, Yusuke; Suga, Masaki; Kido, Masahiro; Yanagimoto, Hiroaki; Toyama, Hirochika; Tokumaru, Sunao; Okimoto, Tomoaki; Terai, Yoshito; Fukumoto, Takumi