The discovery of potent blockers of the canonical transient receptor channels, TRPC3 and TRPC6, based on an anilino-thiazole pharmacophore
基于苯胺基噻唑药效团的典型瞬时受体通道 TRPC3 和 TRPC6 的强效阻断剂的发现
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.5
doi:10.1016/j.bmcl.2013.06.047
David G Washburn, Dennis A Holt, Jason Dodson, Jeff J McAtee, Lamont R Terrell, Linda Barton, Sharada Manns, Anna Waszkiewicz, Christina Pritchard, Dan J Gillie, Dwight M Morrow, Elizabeth A Davenport, Irina M Lozinskaya, Jeffrey Guss, Jonathan B Basilla, Lorena Kallal Negron, Michael Klein, Robert