日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase Inhibition

2-苯基喹啉类化合物通过抑制非结构蛋白13解旋酶发挥抗严重急性呼吸综合征冠状病毒2活性

Cernicchi, Giada; Nizi, Maria Giulia; Emmolo, Roberta; Persoons, Leentje; Laporte, Manon; Jochmans, Dirk; Romeo, Isabella; Pepe, Giacomo; Milite, Ciro; Campiglia, Pietro; Spezzini, Jacopo; Martelli, Alma; Brogi, Simone; Esposito, Francesca; Felicetti, Tommaso; Massari, Serena; Manfroni, Giuseppe; Sabatini, Stefano; Sbardella, Gianluca; Alcaro, Stefano; Neyts, Johan; Corona, Angela; Tramontano, Enzo; De Jonghe, Steven; Tabarrini, Oriana

DNA damage response defects induced by the formation of TDP-43 and mutant FUS cytoplasmic inclusions and their pharmacological rescue.

TDP-43 和突变型 FUS 细胞质内含物的形成引起的 DNA 损伤反应缺陷及其药物挽救。

Modafferi Stefania, Farina Stefania, Esposito Francesca, Brandi Ornella, Di Salvio Michela, Della Valle Ilaria, D'Uva Sara, Scarian Eveljn, Cicio Giada, Riccardi Adelaide, Pisati Federica, Garbelli Anna, Santini Tiziana, Pansarasa Orietta, Morlando Mariangela, D'Ambrosi Nadia, Cozzolino Mauro, Cestra Gianluca, d'Adda di Fagagna Fabrizio, Gioia Ubaldo, Francia Sofia

DROSHA, DICER, and damage-induced long ncRNA control BMI1-dependent transcriptional repression at DNA double-strand break.

DROSHA、DICER 和损伤诱导的长链非编码RNA控制DNA双链断裂处的BMI1依赖性转录抑制。

Esposito Francesca, Capozzo Ilaria, Riccardi Adelaide, Gioia Ubaldo, Modafferi Stefania, Manfredi Letizia, Colantoni Alessio, Tavella Sara, Cabrini Matteo, Iannelli Fabio, di Lillo Alessia, d'Adda di Fagagna Fabrizio, Francia Sofia

N-alkyl and N-benzyl indoles are anti-SARS-CoV-2 agents and nsp13 inhibitors

N-烷基和N-苄基吲哚是抗SARS-CoV-2药物和nsp13抑制剂

Albano, Aurora; Emmolo, Roberta; De Santis, Riccardo; Patacchini, Elisa; Madia, Valentina Noemi; Maloccu, Stefania; Ialongo, Davide; Ruggieri, Giuseppe; Arpacioglu, Merve; Scipione, Luigi; Saccoliti, Francesco; Amatore, Donatella; Grilli, Giorgia; Lista, Florigio; Esposito, Francesca; Tramontano, Enzo; Corona, Angela; Di Santo, Roberto; Costi, Roberta

2-(Trihydroxyphenyl)thienopyrimidinones as Key Scaffolds for Targeting a Novel Allosteric Site of HIV-1 Integrase

2-(三羟基苯基)噻吩并嘧啶酮作为靶向HIV-1整合酶新型变构位点的关键骨架

Tocco, Graziella; Laus, Antonio; Casula, Mattia; Caboni, Pierluigi; Beutler, John A; Tramontano, Enzo; Esposito, Francesca

Cardiac resynchronization therapy in cancer patients with chemotherapy-induced cardiomyopathy: a mini review

化疗诱发心肌病癌症患者的心脏再同步治疗:简要综述

Valzania, Cinzia; Calvi, Valeria; Schirripa, Valentina; Esposito, Francesca; Donnici, Giovanni; Borrello, Francesco; Arestia, Alberto; Sassone, Biagio

Toxicity Assessment of (4Z)-Lachnophyllum and (4Z,8Z)-Matricaria Lactones: Implications for Environmental Safety of Bioherbicides

(4Z)-毛叶菊内酯和(4Z,8Z)-母菊内酯的毒性评估:对生物除草剂环境安全性的影响

Padilla Suarez, Edith Guadalupe; Zorrilla, Jesús G; Spampinato, Marisa; Pannullo, Teresa; Esposito, Francesca; Fernández-Aparicio, Mónica; Libralato, Giovanni; Siciliano, Antonietta; Masi, Marco; Cimmino, Alessio

Dual-Site Inhibition of SARS-CoV-2 RNA-Dependent RNA Polymerase by Small Molecules Able to Block Viral Replication Identified through a Computer-Aided Drug Discovery Approach

通过计算机辅助药物发现方法鉴定出能够阻断SARS-CoV-2 RNA依赖性RNA聚合酶双位点抑制的小分子

Malune, Paolo; Iaconis, Daniela; Manelfi, Candida; Giunta, Stefano; Emmolo, Roberta; Lunghini, Filippo; Paulis, Annalaura; Talarico, Carmine; Corona, Angela; Beccari, Andrea Rosario; Tramontano, Enzo; Esposito, Francesca

Thiol-Reactive or Redox-Active: Revising a Repurposing Screen Led to a New Invalidation Pipeline and Identified a True Noncovalent Inhibitor Against Papain-like Protease from SARS-CoV-2.

硫醇反应性或氧化还原活性:修改重新定位筛选导致新的无效化流程,并鉴定出针对 SARS-CoV-2 木瓜蛋白酶样蛋白酶的真正非共价抑制剂

Kuzikov Maria, Morasso Stefano, Reinshagen Jeanette, Wolf Markus, Monaco Vittoria, Cozzolino Flora, Golič Grdadolnik Simona, Šket Primož, Plavec Janez, Iaconis Daniela, Summa Vincenzo, Corona Angela, Paulis Annalaura, Esposito Francesca, Tramontano Enzo, Monti Maria, Beccari Andrea R, Manelfi Candida, Windshügel Björn, Gribbon Philip, Storici Paola, Zaliani Andrea

Special Issue "Advances in Antiviral Agents Against SARS-CoV-2 and Its Variants" 2nd Edition

特刊“抗SARS-CoV-2及其变种病毒药物研究进展”第二版

Esposito, Francesca