日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Sulfonyl Anthranilic Acid Analogues Display Pan-Serotype Anti-Dengue Activity by Downregulating the Expression of Ribosomal Proteins Encoded by 5'-Terminal Oligopyrimidine Motif-Containing mRNA

磺酰邻氨基苯甲酸类似物通过下调由含5'末端寡嘧啶基序的mRNA编码的核糖体蛋白的表达,表现出泛血清型抗登革热活性。

Gwee, Chin Piaw; Felicetti, Tommaso; Chan, Kitti Wing Ki; Tan, Min Jie Alvin; Bin Mohd Mazlan, Muhammad Danial; Milite, Ciro; Pepe, Giacomo; Sarnari, Chiara; Ng, Xiao Dan; Phoo, Wint Wint; Tan, Jasmine Hwee Yee; Mah, Marcus G; Watanabe, Satoru; Huang, Jing Xiu; Massari, Serena; Tabarrini, Oriana; Sabatini, Stefano; Campiglia, Pietro; Sbardella, Gianluca; Smith, Gavin J D; Alonso, Sylvie; Sun, Alfred Xuyang; Sobota, Radoslaw M; Vasudevan, Subhash G; Manfroni, Giuseppe

2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase Inhibition

2-苯基喹啉类化合物通过抑制非结构蛋白13解旋酶发挥抗严重急性呼吸综合征冠状病毒2活性

Cernicchi, Giada; Nizi, Maria Giulia; Emmolo, Roberta; Persoons, Leentje; Laporte, Manon; Jochmans, Dirk; Romeo, Isabella; Pepe, Giacomo; Milite, Ciro; Campiglia, Pietro; Spezzini, Jacopo; Martelli, Alma; Brogi, Simone; Esposito, Francesca; Felicetti, Tommaso; Massari, Serena; Manfroni, Giuseppe; Sabatini, Stefano; Sbardella, Gianluca; Alcaro, Stefano; Neyts, Johan; Corona, Angela; Tramontano, Enzo; De Jonghe, Steven; Tabarrini, Oriana

In Vitro and In Vivo Investigations into the Potential of Quinazoline and Quinoline Derivatives as NorA Efflux Pump Inhibitors Against Resistant Staphylococcus aureus Strains

体外和体内研究喹唑啉及其衍生物作为NorA外排泵抑制剂对抗耐药金黄色葡萄球菌菌株的潜力

Chandal, Nishtha; Sharma, Nidhi; Cernicchi, Giada; Felicetti, Tommaso; Rondini, Tommaso; Acito, Mattia; Nandanwar, Hemraj; Sabatini, Stefano

NorA Efflux Pump Inhibitors: Expanding SAR Knowledge of Pyrazolo[4,3-c][1,2]benzothiazine 5,5-Dioxide Derivatives

NorA 外排泵抑制剂:扩展吡唑并[4,3-c][1,2]苯并噻嗪 5,5-二氧化物衍生物的构效关系知识

Cernicchi, Giada; Di Gregorio, Alessandra; Felicetti, Tommaso; Rampacci, Elisa; Casari, Giulia; Armeni, Tatiana; Romaldi, Brenda; Zefaj, Ermelinda; Passamonti, Fabrizio; Massari, Serena; Manfroni, Giuseppe; Barreca, Maria Letizia; Tabarrini, Oriana; Vignaroli, Carla; Sabatini, Stefano

Broad-Spectrum Antiviral Activity of Pyridobenzothiazolone Analogues Against Respiratory Viruses.

吡啶并苯并噻唑啉酮类似物对呼吸道病毒的广谱抗病毒活性

Feyles Elisa, Felicetti Tommaso, Arduino Irene, Rittà Massimo, Civra Andrea, Muratori Luisa, Raimondo Stefania, Lembo David, Manfroni Giuseppe, Donalisio Manuela

New Pyridobenothiazolone Derivatives Display Nanomolar Pan-Serotype Anti-Dengue Virus Activity.

新型吡啶并噻唑啉酮衍生物显示出纳摩尔级泛血清型抗登革病毒活性

Felicetti Tommaso, Gwee Chin Piaw, Chan Kitti Wing Ki, Pepe Giacomo, Milite Ciro, Campiglia Pietro, Watanabe Satoru, Mazlan Muhammad Danial Bin Mohd, Sabatini Stefano, Massari Serena, Tabarrini Oriana, Sbardella Gianluca, Vasudevan Subhash G, Manfroni Giuseppe

Fighting Antimicrobial Resistance: Insights on How the Staphylococcus aureus NorA Efflux Pump Recognizes 2-Phenylquinoline Inhibitors by Supervised Molecular Dynamics (SuMD) and Molecular Docking Simulations

对抗抗菌素耐药性:通过监督分子动力学 (SuMD) 和分子对接模拟揭示金黄色葡萄球菌 NorA 外排泵如何识别 2-苯基喹啉抑制剂

Palazzotti, Deborah; Felicetti, Tommaso; Sabatini, Stefano; Moro, Stefano; Barreca, Maria Letizia; Sturlese, Mattia; Astolfi, Andrea

Inhibition of Staphylococcus pseudintermedius Efflux Pumps by Using Staphylococcus aureus NorA Efflux Pump Inhibitors

利用金黄色葡萄球菌NorA外排泵抑制剂抑制中间葡萄球菌外排泵

Rampacci, Elisa; Felicetti, Tommaso; Cernicchi, Giada; Stefanetti, Valentina; Sabatini, Stefano; Passamonti, Fabrizio

Biofunctionalization of Poly(lactide-co-glycolic acid) Using Potent NorA Efflux Pump Inhibitors Immobilized on Nanometric Alpha-Zirconium Phosphate to Reduce Biofilm Formation

利用固定在纳米级α-磷酸锆上的强效NorA外排泵抑制剂对聚乳酸-羟基乙酸共聚物进行生物功能化,以减少生物膜的形成

Pica, Monica; Messere, Nicla; Felicetti, Tommaso; Sabatini, Stefano; Pietrella, Donatella; Nocchetti, Morena

Modulating microRNA Processing: Enoxacin, the Progenitor of a New Class of Drugs

调控microRNA加工:依诺沙星,一类新型药物的先驱

Felicetti, Tommaso; Cecchetti, Violetta; Manfroni, Giuseppe