日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A STAT3 degrader demonstrates efficacy in venetoclax resistant acute myeloid leukemia

STAT3降解剂在维奈托克耐药的急性髓系白血病中显示出疗效

Chakraborty, Samarpana; Morganti, Claudia; Zaldana, Kimberly; Rivera Pena, Bianca; Zhang, Hui; Verma, Divij; Gitego, Nadege; Ma, Feiyang; Aluri, Srinivas; Pradhan, Kith; Gordon-Mitchell, Shanisha; Mantzaris, Ioannis; Goldfinger, Mendel; Feldman, Eric; Gritsman, Kira; Shi, Yang; Hubner, Stefan; Qiu, Yi Hua; Brown, Brandon D; Khasawneh, Abdullah; Skwarska, Anna; de Camargo Magalhães, Eduardo Sabino; Verma, Amit; Konopleva, Marina; Tabe, Yoko; Gavathiotis, Evripidis; Colla, Simona; Gollob, Jared; Dey, Joyoti; Kornblau, Steven M; Koralov, Sergei B; Ito, Keisuke; Shastri, Aditi

RAS Mutation-Specific Responses to Paralog- and State-Selective RAS Inhibitors.

RAS 突变特异性反应对旁系同源和状态选择性 RAS 抑制剂的反应。

Baars Beau, Orive-Ramos Ana, Emmett Matthew J, Gaire Bijaya, Desaunay Mathieu, Kou Ziyue, Li Guangyan, Adamopoulos Christos, Aaronson Stuart A, Wang Shaomeng, Sellers William R, Martin Tiphaine, Gavathiotis Evripidis, Poulikakos Poulikos I

Resistance mechanisms and therapeutic strategies of CDK4 and CDK6 kinase targeting in cancer

癌症中 CDK4 和 CDK6 激酶靶向治疗的耐药机制和治疗策略

Asciolla, James J; Wu, Xuewei; Adamopoulos, Christos; Gavathiotis, Evripidis; Poulikakos, Poulikos I

Small molecule OPA1 inhibitors amplify cytochrome c release and reverse cancer cells resistance to Bcl-2 inhibitors

小分子OPA1抑制剂可增强细胞色素c的释放,并逆转癌细胞对Bcl-2抑制剂的耐药性。

Anna Pellattiero,Charlotte Quirin,Federico Magrin,Mattia Sturlese,Alberto Fracasso,Nikolaos Biris,Stéphanie Herkenne,Laura Cendron,Evripidis Gavathiotis,Stefano Moro,Andrea Mattarei,Luca Scorrano

Defective chaperone-mediated autophagy in the retinal pigment epithelium of age-related macular degeneration patients

年龄相关性黄斑变性患者视网膜色素上皮细胞中分子伴侣介导的自噬缺陷

Juan Ignacio Jiménez-Loygorri ,Peng Shang ,Ibrahim Bayramoglu ,Raquel Gómez-Sintes ,Adrián Martín-Segura ,Helena Ambrosino ,Johnson Hoang ,Antonio Díaz ,Zhaohui Geng ,Evripidis Gavathiotis ,James R Dutton ,Jörn Dengjel ,Ana Maria Cuervo ,Deborah A Ferrington ,Patricia Boya

Small molecule disruption of RARα/NCoR1 interaction inhibits chaperone-mediated autophagy in cancer

小分子干扰 RARα/NCoR1 相互作用可抑制癌症中分子伴侣介导的自噬。

Mericka McCabe ,Rajanya Bhattacharyya ,Rebecca Sereda ,Olaya Santiago-Fernández ,Rabia R Khawaja ,Antonio Diaz ,Kristen Lindenau ,Deniz Gulfem Ozturk ,Thomas P Garner ,Simone Sidoli ,Ana Maria Cuervo ,Evripidis Gavathiotis

Quiescent OXPHOS-High Triple-Negative Breast Cancer Cells That Persist After Chemotherapy Depend on BCL-XL for Survival

化疗后仍能存活的静止期高氧化磷酸化三阴性乳腺癌细胞依赖BCL-XL生存

Andrzejewski, Slawomir; Winter, Marie; Encarnacao Garcia, Leandro; Akinrinmade, Olusiji; Madeira Marques, Francisco; Zacharioudakis, Emmanouil; Skwarska, Anna; Aguirre-Ghiso, Julio; Konopleva, Marina; Zheng, Guangrong; Fineberg, Susan A; Zhou, Daohong; Gavathiotis, Evripidis; Wang, Tao; Dhimolea, Eugen

Quiescent OXPHOS-high triple-negative breast cancer cells that persist after chemotherapy depend on BCL-XL for survival

化疗后仍然存在的静止期、OXPHOS高表达的三阴性乳腺癌细胞依赖BCL-XL生存。

Andrzejewski, Slawomir; Winter, Marie; Garcia, Leandro Encarnacao; Akinrinmade, Olusiji; Marques, Francisco D M; Zacharioudakis, Emmanouil; Skwarska, Anna; Aguirre-Ghiso, Julio; Konopleva, Marina; Zheng, Guangrong; Fineberg, Susan; Zhou, Daohong; Gavathiotis, Evripidis; Wang, Tao; Dhimolea, Eugen

Author Correction: Apoptotic stress causes mtDNA release during senescence and drives the SASP

作者更正:细胞凋亡应激导致衰老过程中线粒体DNA释放,并驱动衰老相关分泌表型(SASP)。

Victorelli, Stella; Salmonowicz, Hanna; Chapman, James; Martini, Helene; Vizioli, Maria Grazia; Riley, Joel S; Cloix, Catherine; Hall-Younger, Ella; Machado Espindola-Netto, Jair; Jurk, Diana; Lagnado, Anthony B; Sales Gomez, Lilian; Farr, Joshua N; Saul, Dominik; Reed, Rebecca; Kelly, George; Eppard, Madeline; Greaves, Laura C; Dou, Zhixun; Pirius, Nicholas; Szczepanowska, Karolina; Porritt, Rebecca A; Huang, Huijie; Huang, Timothy Y; Mann, Derek A; Masuda, Claudio Akio; Khosla, Sundeep; Dai, Haiming; Kaufmann, Scott H; Zacharioudakis, Emmanouil; Gavathiotis, Evripidis; LeBrasseur, Nathan K; Lei, Xue; Sainz, Alva G; Korolchuk, Viktor I; Adams, Peter D; Shadel, Gerald S; Tait, Stephen W G; Passos, João F

Alzheimer's disease-linked risk alleles elevate microglial cGAS-associated senescence and neurodegeneration in a tauopathy model.

阿尔茨海默病相关风险等位基因在 tau 蛋白病模型中加剧小胶质细胞 cGAS 相关的衰老和神经退行性变

Carling Gillian K, Fan Li, Foxe Nessa R, Norman Kendra, Wong Man Ying, Zhu Daphne, Corona Carlo, Razzoli Agnese, Yu Fangmin, Yarahmady Allan, Ye Pearly, Chen Hao, Huang Yige, Amin Sadaf, Sereda Rebecca, Lopez-Lee Chloe, Zacharioudakis Emmanouil, Chen Xiaoying, Xu Jielin, Cheng Feixiong, Gavathiotis Evripidis, Cuervo Ana Maria, Holtzman David M, Mok Sue-Ann, Sinha Subhash C, Sidoli Simone, Ratan Rajiv R, Luo Wenjie, Gong Shiaoching, Gan Li