First-in-class inhibitors of Nsp15 endoribonuclease of SARS-CoV-2: Modeling, synthesis, and enzymatic assay of thiazolidinedione and rhodanine analogs
SARS-CoV-2 Nsp15 核糖核酸内切酶的首创抑制剂:噻唑烷二酮和罗丹宁类似物的建模、合成和酶活性测定
期刊:Journal of Biological Chemistry
影响因子:3.9
doi:10.1016/j.jbc.2025.110409
Mehyar, Nimer; Samman, Nosaibah; Al Gheribi, Shatha; Mashhour, Abdullah; Chan, Pearl; Al-Kaysi, Rabih O; Perlman, Stanley; Boudjelal, Mohamed; Islam, Imadul