日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting transcription factors through an IMiD independent zinc finger domain.

通过不依赖于IMiD的锌指结构域靶向转录因子

Liu Bee Hui, Liu Miao, Radhakrishnan Sridhar, Dai Meng-Yuan, Jaladanki Chaitanya Kumar, Gao Chong, Tang Jing Ping, Kumari Kalpana, Go Mei Lin, Vu Kim Anh L, Kwon Junsu, Seo Hyuk-Soo, Song Kijun, Tian Xi, Feng Li, Tan Justin L, Melkonian Arek V, Liu Zhaoji, Wulf Gerburg, Arthanari Haribabu, Qi Jun, Dhe-Paganon Sirano, Clohessy John G, Choong Yeu Khai, Sivaraman J, Fan Hao, Tenen Daniel G, Chai Li

A potent phenylalkylamine disrupts mycobacterial membrane bioenergetics and augments bactericidal activity of bedaquiline.

一种强效的苯烷基胺可破坏分枝杆菌膜生物能量学,并增强贝达喹啉的杀菌活性

Phua Zheng Yen, Li Ming, Ali Azhar, Cheong Cedric Cheng Sheng, Goh Kai Jie, Seto Marcus Yi Kang, Ng Amos Shi Ying, Sarathy Jickky Palmae, Goh Boon Cher, Go Mei Lin, Chui Wai Keung, Dick Thomas, Lam Yulin

PROTAC antibiotics: the time is now

PROTAC抗生素:时机已到

Sarathy, Jickky Palmae; Aldrich, Courtney C; Go, Mei-Lin; Dick, Thomas

Redox Cycling Dioxonaphthoimidazoliums Disrupt Iron Homeostasis in Mycobacterium bovis Bacillus Calmette-Guérin

二氧萘并咪唑类化合物的氧化还原循环会破坏牛分枝杆菌和卡介苗中的铁稳态。

Li, Ming; Yamada, Yoshiyuki; Rodriguez, G Marcela; Dick, Thomas; Go, Mei Lin

Alkyltriphenylphosphonium turns naphthoquinoneimidazoles into potent membrane depolarizers against mycobacteria

烷基三苯基膦可将萘醌咪唑转化为对抗分枝杆菌的强效膜去极化剂

Fridianto, Kevin Timothy; Gunawan, Gregory Adrian; Hards, Kiel; Sarathy, Jickky Palmae; Cook, Gregory M; Dick, Thomas; Go, Mei-Lin; Lam, Yulin

Functionalized Dioxonaphthoimidazoliums: A Redox Cycling Chemotype with Potent Bactericidal Activities against Mycobacterium tuberculosis

功能化二氧萘并咪唑鎓:一种具有强效抗结核分枝杆菌杀菌活性的氧化还原循环化学型

Fridianto, Kevin T; Li, Ming; Hards, Kiel; Negatu, Dereje A; Cook, Gregory M; Dick, Thomas; Lam, Yulin; Go, Mei-Lin

Effects of Antimalarial Drugs on Neuroinflammation-Potential Use for Treatment of COVID-19-Related Neurologic Complications

抗疟药对神经炎症的影响——治疗新冠肺炎相关神经系统并发症的潜在用途

Ong, Wei-Yi; Go, Mei-Lin; Wang, De-Yun; Cheah, Irwin Kee-Mun; Halliwell, Barry

Amide-Amine Replacement in Indole-2-carboxamides Yields Potent Mycobactericidal Agents with Improved Water Solubility

吲哚-2-甲酰胺中的酰胺-胺取代可产生具有更高水溶性的强效杀分枝杆菌剂

Tan, Yu Jia; Li, Ming; Gunawan, Gregory Adrian; Nyantakyi, Samuel Agyei; Dick, Thomas; Go, Mei-Lin; Lam, Yulin

Rifabutin Suppresses Inducible Clarithromycin Resistance in Mycobacterium abscessus by Blocking Induction of whiB7 and erm41

利福布汀通过阻断 whiB7 和 erm41 的诱导来抑制脓肿分枝杆菌中诱导型克拉霉素耐药性

Aziz, Dinah Binte; Go, Mei Lin; Dick, Thomas

Resistance against Membrane-Inserting MmpL3 Inhibitor through Upregulation of MmpL5 in Mycobacterium tuberculosis

结核分枝杆菌通过上调 MmpL5 产生对膜插入 MmpL3 抑制剂的耐药性

Li, Ming; Nyantakyi, Samuel Agyei; Go, Mei-Lin; Dick, Thomas