日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In Vitro and In Vivo Characterization of Novel Cathelicidin-Based Peptides with Antimicrobial Activity Against Pseudomonas aeruginosa.

体外和体内表征新型抗菌肽对铜绿假单胞菌的抗菌活性

Moreno-Morales Javier, Martín-Vilardell Núria, Guardiola Salvador, Vila-Farrés Xavier, Cebrero Tania, Babić Marko, Ballesté-Delpierre Clara, Kalafatović Daniela, Giralt Ernest, Pachón-Ibañez María Eugenia, Vila Jordi

Angiotensin-(1-9) Retro-Enantiomer Peptide With Cardioprotective Activity

具有心脏保护活性的血管紧张素-(1-9)逆对映体肽

Flores, Yvo; Zapata-Torres, Gerald; Nuñez, Agustín; Matthies, Douglas J; Alemán, Larissa; Hernández-Fuentes, Carolina; Sánchez, Gina; Araya, Eyleen; Guzman, Fanny; Pedrozo, Zully; Guardiola, Salvador; Varese, Mónica; Giralt, Ernest; Maslov, Ivan; Del Borgo, Mark; Widdop, Robert E; Valdebenito, Silvana; Eugenin, Eliseo A; Chiong, Mario; Hill, Joseph A; Ocaranza, María Paz; Kogan, Marcelo J; Lavandero, Sergio

In vivo photocontrol of orexin receptors with a nanomolar light-regulated analogue of orexin-B

利用纳摩尔级光调控的食欲素B类似物对食欲素受体进行体内光控。

Prischich, Davia; Sortino, Rosalba; Gomila-Juaneda, Alexandre; Matera, Carlo; Guardiola, Salvador; Nepomuceno, Diane; Varese, Monica; Bonaventure, Pascal; de Lecea, Luis; Giralt, Ernest; Gorostiza, Pau

Target-templated de novo design of macrocyclic d-/l-peptides: discovery of drug-like inhibitors of PD-1

以靶标为模板从头设计大环d-/l-肽:发现PD-1的类药抑制剂

Guardiola, Salvador; Varese, Monica; Roig, Xavier; Sánchez-Navarro, Macarena; García, Jesús; Giralt, Ernest

Small molecule inhibits α-synuclein aggregation, disrupts amyloid fibrils, and prevents degeneration of dopaminergic neurons

小分子抑制α-突触核蛋白聚集,破坏淀粉样蛋白原纤维,并防止多巴胺能神经元退化。

Pujols, Jordi; Peña-Díaz, Samuel; Lázaro, Diana F; Peccati, Francesca; Pinheiro, Francisca; González, Danilo; Carija, Anita; Navarro, Susanna; Conde-Giménez, María; García, Jesús; Guardiola, Salvador; Giralt, Ernest; Salvatella, Xavier; Sancho, Javier; Sodupe, Mariona; Outeiro, Tiago Fleming; Dalfó, Esther; Ventura, Salvador