日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeted degradation of CDK9 potently disrupts the MYC-regulated network.

靶向降解 CDK9 可有效破坏 MYC 调控网络

Toure Mohammed A, Motoyama Keisuke, Xiang Yichen, Urgiles Julie, Kabinger Florian, Koglin Ann-Sophie, Iyer Ramya S, Gagnon Kaitlyn, Kumar Amruth, Ojeda Samuel, Harrison Drew A, Rees Matthew G, Roth Jennifer A, Ott Christopher J, Schiavoni Richard, Whittaker Charles A, Levine Stuart S, White Forest M, Calo Eliezer, Richters Andre, Koehler Angela N

Structure-Guided Design of ISOX-DUAL-Based Degraders Targeting BRD4 and CBP/EP300: A Case of Degrader Collapse.

基于 ISOX-DUAL 的结构导向降解剂设计:针对 BRD4 和 CBP/EP300 的降解剂崩溃案例

Edmonds Anthony K, Balourdas Dimitrios-Ilias, Marsh Graham P, Felix Robert, Brasher Bradley, Cooper Jeff, Graber-Feesl Cari, Kollareddy Madhu, Malik Karim, Stewart Helen, Chevassut Timothy J T, Lineham Ella, Morley Simon, Fedorov Oleg, Bennett James, Rajasekaran Mohan B, Ojeda Samuel, Harrison Drew A, Ott Christopher J, Joerger Andreas C, Maple Hannah J, Spencer John

Development of p300-targeting degraders with enhanced selectivity and onset of degradation.

开发具有增强选择性和更快降解速度的p300靶向降解剂

Marsh Graham P, Cooper Mark S, Goggins Sean, Reynolds Stephen J, Wheeler Dean F, Cresser-Brown Joel O, Arnold Robert E, Babcock Emily G, Hughes Gareth, Bosnakovski Darko, Kyba Michael, Ojeda Samuel, Harrison Drew A, Ott Christopher J, Maple Hannah J