日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Constitutive activity of an atypical chemokine receptor revealed by inverse agonistic nanobodies

反向激动性纳米抗体揭示非典型趋化因子受体的组成型活性

Perez Almeria, Claudia V; Otun, Omolade; Schlimgen, Roman; Lamme, Thomas D; Di Niro, Lotte; Crudden, Caitrin; Bebelman, Jan Paul; Youssef, Noureldine; Musli, Lejla; Jenjak, Shawn; Bobkov, Vladimir; Drube, Julia; Hoffmann, Carsten; Volkman, Brian F; Granier, Sébastien; Bechara, Cherine; Siderius, Marco; Heukers, Raimond; Schafer, Christopher T; Smit, Martine J

Disruption of constitutive CXCR4 oligomers impairs oncogenic properties in lymphoid neoplasms.

CXCR4 寡聚体的组成破坏会损害淋巴瘤的致癌特性

Mobach Simon, Bergkamp Nick D, Ma Ziliang, Haselager Marco V, Anbuhl Stephanie M, Jurriens Daphne, van den Bor Jelle, Wang Ziming, Crudden Caitrin, Roos Jamie L, Perez Almeria Claudia V, Boergonje Rick A, Lohse Martin J, Bosma Reggie, Eldering Eric, Siderius Marco, Wu Wei, Spaargaren Marcel, Tonino Sanne H, Kater Arnon P, Smit Martine J, Heukers Raimond

TR-FRET between engineered nanobodies reveals the existence of endogenous CXCR4 oligomers

利用工程纳米抗体之间的时间分辨荧光共振能量转移(TR-FRET)技术揭示了内源性CXCR4寡聚体的存在。

Heuninck, Joyce; Bobkov, Vladimir; Grison, Claire M; Fumagalli, Amos; Lescuyer, Mathias; Otun, Omolade; Bechara, Cherine; Lamarque, Laurent; Trinquet, Eric; Bachelerie, Françoise; Marin, Philippe; Mouillac, Bernard; Granier, Sébastien; van der Woning, Bas; de Haard, Hans; Smit, Martine J; Heukers, Raimond; Durroux, Thierry

Genetic Engineering of VHH Antibody Fragments for Efficient Site-Specific Conjugation to Polysaccharides.

利用基因工程技术对VHH抗体片段进行高效位点特异性偶联,以与多糖结合

Zhong Lin, Morshuis Lisanne C M, Koerselman Michelle, Memelink Angela, Kolecka Anna, Heukers Raimond, Verrips Theo, Karperien Marcel, Zoetebier Bram

Plasma membrane rather than endosomal Gq signaling drives transcriptional activity by the viral chemokine receptor US28 in glioblastoma

在胶质母细胞瘤中,病毒趋化因子受体US28的转录活性是由质膜而非内体Gq信号传导驱动的。

Daly, Carole; Wright, Adam; Heukers, Raimond; McKee, Chloe M; Coll, Rebecca C; Evergren, Emma; Smit, Martine J; Thomsen, Alex R B; Plouffe, Bianca

Structural basis for selectivity and antagonism in extracellular GPCR-nanobodies

细胞外GPCR纳米抗体选择性和拮抗作用的结构基础

Roman R Schlimgen ,Francis C Peterson ,Raimond Heukers ,Martine J Smit ,John D McCorvy ,Brian F Volkman

Inhibition of HIV-1 replication by nanobodies targeting tetraspanin CD9

靶向四跨膜蛋白CD9的纳米抗体抑制HIV-1复制

Jeffrey C Umotoy ,Pascal Z Kroon ,Shirley Man ,Karel A van Dort ,Tugba Atabey ,Angela I Schriek ,Gillian Dekkers ,Elena Herrera-Carrillo ,Teunis B H Geijtenbeek ,Raimond Heukers ,Neeltje A Kootstra ,Marit J van Gils ,Steven W de Taeye

Constitutive activity of an atypical chemokine receptor revealed by inverse agonistic nanobodies

反向激动剂纳米抗体揭示非典型趋化因子受体的组成活性

Claudia V Perez Almeria, Omolade Otun, Roman Schlimgen, Thomas D Lamme, Caitrin Crudden, Noureldine Youssef, Lejla Musli, Shawn Jenjak, Vladimir Bobkov, Julia Drube, Carsten Hoffmann, Brian F Volkman, Sébastien Granier, Cherine Bechara, Marco Siderius, Raimond Heukers, Christopher T Schafer, Martine

Molecular characterization of the CXCR4 / CXCR7 axis in germ cell tumors and its targetability using nanobody-drug-conjugates

生殖细胞肿瘤中CXCR4/CXCR7轴的分子特征及其纳米抗体-药物偶联靶向性研究

Wakileh, Gamal A; Bierholz, Philipp; Kotthoff, Mara; Skowron, Margaretha A; Bremmer, Felix; Stephan, Alexa; Anbuhl, Stephanie M; Heukers, Raimond; Smit, Martine J; Ströbel, Philipp; Nettersheim, Daniel

NanoB2 to monitor interactions of ligands with membrane proteins by combining nanobodies and NanoBRET

NanoB2 通过结合纳米抗体和 NanoBRET 来监测配体与膜蛋白的相互作用

Jelle van den Bor, Nick D Bergkamp, Stephanie M Anbuhl, Françoise Dekker, Dehan Comez, Claudia V Perez Almeria, Reggie Bosma, Carl W White, Laura E Kilpatrick, Stephen J Hill, Marco Siderius, Martine J Smit, Raimond Heukers