Discovery and Characterization of SY-1365, a Selective, Covalent Inhibitor of CDK7
SY-1365(CDK7 选择性共价抑制剂)的发现和表征
期刊:Cancer Research
影响因子:12.5
doi:10.1158/0008-5472.CAN-19-0119
Shanhu Hu, Jason J Marineau, Nisha Rajagopal, Kristin B Hamman, Yoon Jong Choi, Darby R Schmidt, Nan Ke, Liv Johannessen, Michael J Bradley, David A Orlando, Sydney R Alnemy, Yixuan Ren, Stephane Ciblat, Dana K Winter, Anzhelika Kabro, Kevin T Sprott, J Graeme Hodgson, Christian C Fritz, John P Caru