日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

DUSP4 protects BRAF- and NRAS-mutant melanoma from oncogene overdose through modulation of MITF

DUSP4 通过调节 MITF 来保护 BRAF 和 NRAS 突变型黑色素瘤免受癌基因过载的影响。

Nuria Gutierrez-Prat ,Hedwig L Zuberer ,Luca Mangano ,Zahra Karimaddini ,Luise Wolf ,Stefka Tyanova ,Lisa C Wellinger ,Daniel Marbach ,Vera Griesser ,Piergiorgio Pettazzoni ,James R Bischoff ,Daniel Rohle ,Chiara Palladino ,Igor Vivanco

A systematic molecular and pharmacologic evaluation of AKT inhibitors reveals new insight into their biological activity

对AKT抑制剂进行系统的分子和药理学评价,揭示了其生物活性的新见解。

Eleftherios Kostaras # ,Teresa Kaserer # ,Glorianne Lazaro ,Sara Farrah Heuss ,Aasia Hussain ,Pedro Casado ,Angela Hayes ,Cihangir Yandim ,Nicolaos Palaskas ,Yi Yu ,Brian Schwartz ,Florence Raynaud ,Yuen-Li Chung ,Pedro R Cutillas ,Igor Vivanco

EGFR feedback-inhibition by Ran-binding protein 6 is disrupted in cancer

癌症中,Ran结合蛋白6对EGFR的反馈抑制作用遭到破坏。

Barbara Oldrini ,Wan-Ying Hsieh ,Hediye Erdjument-Bromage ,Paolo Codega ,Maria Stella Carro ,Alvaro Curiel-García ,Carl Campos ,Maryam Pourmaleki ,Christian Grommes ,Igor Vivanco ,Daniel Rohle ,Craig M Bielski ,Barry S Taylor ,Travis J Hollmann ,Marc Rosenblum ,Paul Tempst ,John Blenis ,Massimo Squatrito ,Ingo K Mellinghoff

IQGAP1 controls tight junction formation through differential regulation of claudin recruitment

IQGAP1通过差异调节紧密连接的募集来控制紧密连接的形成

Barbara E Tanos, Andres E Perez Bay, Susana Salvarezza, Igor Vivanco, Ingo Mellinghoff, Mahasin Osman, David B Sacks, Enrique Rodriguez-Boulan

A kinase-independent function of AKT promotes cancer cell survival

AKT 的激酶非依赖性功能促进癌细胞存活

Igor Vivanco, Zhi C Chen, Barbara Tanos, Barbara Oldrini, Wan-Ying Hsieh, Nicolas Yannuzzi, Carl Campos, Ingo K Mellinghoff

Differential sensitivity of glioma- versus lung cancer-specific EGFR mutations to EGFR kinase inhibitors

胶质瘤和肺癌特异性 EGFR 突变对 EGFR 激酶抑制剂的不同敏感性

Igor Vivanco, H Ian Robins, Daniel Rohle, Carl Campos, Christian Grommes, Phioanh Leia Nghiemphu, Sara Kubek, Barbara Oldrini, Milan G Chheda, Nicolas Yannuzzi, Hui Tao, Shaojun Zhu, Akio Iwanami, Daisuke Kuga, Julie Dang, Alicia Pedraza, Cameron W Brennan, Adriana Heguy, Linda M Liau, Frank Lieberm

Glucose deprivation activates a metabolic and signaling amplification loop leading to cell death

葡萄糖缺乏会激活代谢和信号放大回路,导致细胞死亡

Nicholas A Graham, Martik Tahmasian, Bitika Kohli, Evangelia Komisopoulou, Maggie Zhu, Igor Vivanco, Michael A Teitell, Hong Wu, Antoni Ribas, Roger S Lo, Ingo K Mellinghoff, Paul S Mischel, Thomas G Graeber