日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A Dynamic and Combinatorial Histone Code Drives Malaria Parasite Asexual and Sexual Development

动态和组合组蛋白代码驱动疟原虫无性和有性发育

Hilde von Grüning, Mariel Coradin, Mariel R Mendoza, Janette Reader, Simone Sidoli, Benjamin A Garcia, Lyn-Marié Birkholtz

Semi-Synthetic Analogues of Cryptolepine as a Potential Source of Sustainable Drugs for the Treatment of Malaria, Human African Trypanosomiasis, and Cancer

半合成 Cryptolepine 类似物可作为治疗疟疾、非洲人类锥虫病和癌症的可持续药物的潜在来源

Yabalu Z Abacha, Arnold Donkor Forkuo, Stephen Y Gbedema, Nimisha Mittal, Sabine Ottilie, Frances Rocamora, Elizabeth A Winzeler, Donelly A van Schalkwyk, John M Kelly, Martin C Taylor, Janette Reader, Lyn-Marie Birkholtz, David R Lisgarten, Jeremy K Cockcroft, John N Lisgarten, Rex A Palmer, Rosema

New Transmission-Selective Antimalarial Agents through Hit-to-Lead Optimization of 2-([1,1'-Biphenyl]-4-carboxamido)benzoic Acid Derivatives

通过对 2-([1,1'-联苯]-4-甲酰胺基)苯甲酸衍生物进行先导化合物优化,开发出新型选择性传播抗疟药

Janette Reader, Daniel F L Opperman, Mariëtte E van der Watt, Anjo Theron, Meta Leshabane, Shanté da Rocha, Jonathan Turner, Kathleen Garrabrant, Ivett Piña, Catherine Mills, Patrick M Woster, Lyn-Marié Birkholtz

The ecdysone receptor regulates several key physiological factors in Anopheles funestus

蜕皮激素受体调节不规则按蚊的几个关键生理因素

Surina Maharaj, Elodie Ekoka, Erica Erlank, Luisa Nardini, Janette Reader, Lyn-Marie Birkholtz, Lizette L Koekemoer

Multistage and transmission-blocking targeted antimalarials discovered from the open-source MMV Pandemic Response Box

从开源 MMV 疫情应对箱中发现多阶段和阻断传播的靶向抗疟药

Janette Reader, Mariëtte E van der Watt, Dale Taylor, Claire Le Manach, Nimisha Mittal, Sabine Ottilie, Anjo Theron, Phanankosi Moyo, Erica Erlank, Luisa Nardini, Nelius Venter, Sonja Lauterbach, Belinda Bezuidenhout, Andre Horatscheck, Ashleigh van Heerden, Natalie J Spillman, Anne N Cowell, Jessic

H3K36 methylation reprograms gene expression to drive early gametocyte development in Plasmodium falciparum

H3K36甲基化重新编程基因表达以驱动恶性疟原虫早期配子体发育

Jessica Connacher, Gabrielle A Josling, Lindsey M Orchard, Janette Reader, Manuel Llinás, Lyn-Marié Birkholtz

Naphthylisoquinoline alkaloids, validated as hit multistage antiplasmodial natural products

萘异喹啉生物碱,被证实为热门的多级抗疟原虫天然产物

Phanankosi Moyo, William Shamburger, Mariëtte E van der Watt, Janette Reader, Ana Carolina C de Sousa, Timothy J Egan, Vinesh J Maharaj, Gerhard Bringmann, Lyn-Marie Birkholtz

Optimal 10-Aminoartemisinins With Potent Transmission-Blocking Capabilities for New Artemisinin Combination Therapies-Activities Against Blood Stage P. falciparum Including Pf KI3 C580Y Mutants and Liver Stage P. berghei Parasites

具有强效传播阻断能力的最佳 10 氨基青蒿素,可用于新型青蒿素联合疗法 - 针对血液阶段恶性疟原虫(包括 Pf KI3 C580Y 突变体)和肝脏阶段伯氏疟原虫寄生虫的活性

Ho Ning Wong, Vivian Padín-Irizarry, Mariëtte E van der Watt, Janette Reader, Wilna Liebenberg, Lubbe Wiesner, Peter Smith, Korina Eribez, Elizabeth A Winzeler, Dennis E Kyle, Lyn-Marie Birkholtz, Dina Coertzen, Richard K Haynes

Hierarchical transcriptional control regulates Plasmodium falciparum sexual differentiation

分级转录控制调控恶性疟原虫性别分化

Riëtte van Biljon, Roelof van Wyk, Heather J Painter, Lindsey Orchard, Janette Reader, Jandeli Niemand, Manuel Llinás, Lyn-Marie Birkholtz

Discovery of compounds blocking the proliferation of Toxoplasma gondii and Plasmodium falciparum in a chemical space based on piperidinyl-benzimidazolone analogs

基于哌啶基苯并咪唑酮类似物的化学空间中发现阻断弓形虫和恶性疟原虫增殖的化合物

Nadia Saïdani, Cyrille Y Botté, Michael Deligny, Anne-Laure Bonneau, Janette Reader, Ronald Lasselin, Goulven Merer, Alisson Niepceron, Fabien Brossier, Jean-Christophe Cintrat, Bernard Rousseau, Lyn-Marie Birkholtz, Marie-France Cesbron-Delauw, Jean-François Dubremetz, Corinne Mercier, Henri Vial,