日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Combining BET inhibition with SMAC mimetics restricts tumor growth and triggers immune surveillance in preclinical cancer models

在临床前癌症模型中,BET抑制剂与SMAC模拟物联合使用可抑制肿瘤生长并触发免疫监视。

Ksenija Slavic Obradovic ,Florian Ebner ,Artem V Artemov ,Martina Miotto ,Paula-Elena Traexler ,Robin Jacob ,Ha Pham Thi Thanh ,Regina Ruzicka ,Andreas Wernitznig ,Ines Baumann ,Daniel Gerlach ,Maria-Antonietta Impagnatiello ,Salvatore Siena ,Mary Murphy ,Reniqua House ,Ulrich Reiser ,Valeria Santoro ,Johannes Popow ,Sebastian Carotta ,Anke Baum ,Jesse Lipp ,Alberto Bardelli ,Ulrike Tontsch-Grunt ,Mariangela Russo ,Martin Aichinger

Pan-KRAS Inhibitors BI-2493 and BI-2865 Display Potent Antitumor Activity in Tumors with KRAS Wild-type Allele Amplification

泛KRAS抑制剂BI-2493和BI-2865在KRAS野生型等位基因扩增的肿瘤中显示出强大的抗肿瘤活性

Antonio Tedeschi # ,Fiorella Schischlik # ,Francesca Rocchetti # ,Johannes Popow ,Florian Ebner ,Daniel Gerlach ,Antonia Geyer ,Valeria Santoro ,Andrew S Boghossian ,Matthew G Rees ,Melissa M Ronan ,Jennifer A Roth ,Jesse Lipp ,Matthias Samwer ,Michael Gmachl ,Norbert Kraut ,Mark Pearson ,Dorothea Rudolph