日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Human Myelin Spheres for in Vitro Oligodendrocyte Maturation, Myelination and Neurological Disease Modeling.

用于体外少突胶质细胞成熟、髓鞘形成和神经系统疾病建模的人类髓鞘球。

Ahuja Karan, Ramezankhani Roya, Wang Xinyu, Burg Thibaut, Amos Giulia, Neyrinck Katrien, Silva Alessio, Arekatla Geethika, Cassidy Eleanor Eva, Nami Fatemeharefeh, Terryn Joke, Wierda Keimpe, Vints Katlijn, Vandamme Niels, Poovathingal Suresh, Lambrichts Ivo, Swinnen Johannes V, Van Den Bosch Ludo, De Groef Lies, Moons Lieve, Verfaillie Catherine, Neyts Johan, Jochmans Dirk, Chai Yoke Chin

2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase Inhibition

2-苯基喹啉类化合物通过抑制非结构蛋白13解旋酶发挥抗严重急性呼吸综合征冠状病毒2活性

Cernicchi, Giada; Nizi, Maria Giulia; Emmolo, Roberta; Persoons, Leentje; Laporte, Manon; Jochmans, Dirk; Romeo, Isabella; Pepe, Giacomo; Milite, Ciro; Campiglia, Pietro; Spezzini, Jacopo; Martelli, Alma; Brogi, Simone; Esposito, Francesca; Felicetti, Tommaso; Massari, Serena; Manfroni, Giuseppe; Sabatini, Stefano; Sbardella, Gianluca; Alcaro, Stefano; Neyts, Johan; Corona, Angela; Tramontano, Enzo; De Jonghe, Steven; Tabarrini, Oriana

A coronavirus assembly inhibitor that targets the viral membrane protein.

一种针对病毒膜蛋白的冠状病毒组装抑制剂

Laporte Manon, Jochmans Dirk, Bardiot Dorothée, Desmarets Lowiese, Debski-Antoniak Oliver J, Mizzon Giulia, Abdelnabi Rana, Leyssen Pieter, Chiu Winston, Zhang Zhikuan, Nomura Norimichi, Boland Sandro, Ohto Umeharu, Stahl Yannick, Wuyts Jurgen, De Jonghe Steven, Stevaert Annelies, van Hemert Martijn J, Bontes Brenda W, Wanningen Patrick, Groenewold G J Mirjam, Zegar Aneta, Owczarek Katarzyna, Joshi Sanjata, Koukni Mohamed, Arzel Philippe, Klaassen Hugo, Vanherck Jean-Christophe, Vandecaetsbeek Ilse, Cremers Niels, Donckers Kim, Francken Thibault, Van Buyten Tina, Rymenants Jasper, Schepers Joost, Pyrc Krzysztof, Hilgenfeld Rolf, Dubuisson Jean, Bosch Berend-Jan, Van Kuppeveld Frank, Eydoux Cecilia, Decroly Etienne, Canard Bruno, Naesens Lieve, Weynand Birgit, Snijder Eric J, Belouzard Sandrine, Shimizu Toshiyuki, Bartenschlager Ralf, Hurdiss Daniel L, Marchand Arnaud, Chaltin Patrick, Neyts Johan

Structure-Based Optimization of Pyridone α-Ketoamides as Inhibitors of the SARS-CoV-2 Main Protease

基于结构的吡啶酮α-酮酰胺类化合物作为SARS-CoV-2主蛋白酶抑制剂的优化

Akula, Ravi Kumar; El Kilani, Haifa; Metzen, Alina; Röske, Judith; Zhang, Kaixuan; Göhl, Matthias; Arisetti, Nanaji; Marsh, Graham P; Maple, Hannah J; Cooper, Mark S; Karadogan, Burhan; Jochmans, Dirk; Neyts, Johan; Rox, Katharina; Hilgenfeld, Rolf; Brönstrup, Mark

Identification and Exploration of a Series of SARS-Cov‑2 M(Pro) Cyano-Based Inhibitors Revealing Ortho-Substitution Effects within the P3 Biphenyl Group

鉴定和探索一系列SARS-CoV-2 M(Pro)氰基抑制剂,揭示P3联苯基团中的邻位取代效应

Clyde-Allen, Emma; Zmudzinski, Mikołaj; Afsar, Mohammad; James, Ciyana; Nayak, Anindita; Nayak, Digant; Dos Santos Bury, Priscila; Jochmans, Dirk; Neyts, Johann; Scott, Christopher J; Olsen, Shaun K; Drag, Marcin; Williams, Rich

The Combination of GS-441524 (Remdesivir) and Ribavirin Results in a Potent Antiviral Effect Against Human Parainfluenza Virus 3 Infection in Human Airway Epithelial Cell Cultures and in a Mouse Infection Model

GS-441524(瑞德西韦)与利巴韦林联合用药,在人呼吸道上皮细胞培养物和鼠感染模型中,均能有效抑制人副流感病毒3型感染。

Lin, Yuxia; Weynand, Birgit; Zhang, Xin; Laporte, Manon; Jochmans, Dirk; Neyts, Johan

Discovery of orally bioavailable Zika and West Nile Virus antiviral compounds targeting the NS2B-NS3 protease

发现可口服生物利用的寨卡病毒和西尼罗病毒抗病毒化合物,这些化合物靶向NS2B-NS3蛋白酶

Kenton, Nathaniel T; Barr, Haim; Cherepakha, Artem; Coelmont, Lotte; Collard, Caroline; Cousins, David; Davies, Geraint H M; Degtyarenko, Oleksii; Dirksen, Andrew; Elbrecht, Daniel; Fearon, Daren; Gayvert, James; Griffen, Edward; Jochmans, Dirk; Kaptein, Suzanne; Kliatskiy, Pavlo; Kochetkov, Artem; Kordubailo, Mykyta; Lahav, Noa; London, Nir; Maas, Elke; Marples, Peter; Nady, Nataliya; Neyts, Johan; Nguyen, Luong; Ni, Xiaomin; Ogorodnik, Yuliia; Robinson, Matthew C; Simpson, Carolina Turk; Tarabara, Ihor; Tkachenko, Anton; von Delft, Annette; von Delft, Frank; Yakymenko, Oleksandr; Lee, Alpha A

The triple combination of Remdesivir (GS-441524), Molnupiravir and Ribavirin is highly efficient in inhibiting coronavirus replication in human nasal airway epithelial cell cultures and in a hamster infection model

瑞德西韦(GS-441524)、莫努匹拉韦和利巴韦林的三联疗法能高效抑制人鼻腔气道上皮细胞培养物和仓鼠感染模型中的冠状病毒复制。

Do, Thuc Nguyen Dan; Abdelnabi, Rana; Boda, Bernadett; Constant, Samuel; Neyts, Johan; Jochmans, Dirk

Nirmatrelvir-resistant SARS-CoV-2 is efficiently transmitted in female Syrian hamsters and retains partial susceptibility to treatment.

对尼马替利韦耐药的 SARS-CoV-2 能在雌性叙利亚仓鼠中有效传播,并且对治疗仍保持部分敏感性

Abdelnabi Rana, Jochmans Dirk, Donckers Kim, Trüeb Bettina, Ebert Nadine, Weynand Birgit, Thiel Volker, Neyts Johan

Azapeptide activity-based probes for the SARS-CoV-2 main protease enable visualization of inhibition in infected cells

基于氮杂肽活性的SARS-CoV-2主蛋白酶探针能够可视化感染细胞中的抑制情况。

Vanhoutte, Roeland; Barniol-Xicota, Marta; Chiu, Winston; Vangeel, Laura; Jochmans, Dirk; De Jonghe, Steven; Zidane, Hadeer; Barr, Haim M; London, Nir; Neyts, Johan; Verhelst, Steven H L