日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Pan-TEAD Inhibitors That Disrupt YAP-TEAD Interaction as a Potential Therapy for Gastric Cancers and Mutant KRAS and EGFR Lung Cancers

发现可破坏YAP-TEAD相互作用的泛TEAD抑制剂,有望成为胃癌以及KRAS和EGFR突变型肺癌的潜在疗法

Kumar, Ramesh; Thian, Joanne; Toh, Joel D W; Farzana, Noorul; Sun, Jialin; Kang, CongBao; Low, Suet Mei Crystal; Wee, Sheena; Lim, Zijie; Gunaratne, Jayantha; Loh, Hui Mun; Kannan, Srinivasaraghavan; Verma, Chandra S; Chakraborty, Sayan; Hong, Wanjin

Author Correction: Design-rules for stapled peptides with in vivo activity and their application to Mdm2/X antagonists

作者更正:具有体内活性的肽链设计规则及其在 Mdm2/X 拮抗剂中的应用

Chandramohan, Arun; Josien, Hubert; Yuen, Tsz Ying; Duggal, Ruchia; Spiegelberg, Diana; Yan, Lin; Juang, Yu-Chi Angela; Ge, Lan; Aronica, Pietro G; Kaan, Hung Yi Kristal; Lim, Yee Hwee; Peier, Andrea; Sherborne, Brad; Hochman, Jerome; Lin, Songnian; Biswas, Kaustav; Nestor, Marika; Verma, Chandra S; Lane, David P; Sawyer, Tomi K; Garbaccio, Robert; Henry, Brian; Kannan, Srinivasaraghavan; Brown, Christopher J; Johannes, Charles W; Partridge, Anthony W

Conserved leucine-rich repeat proteins in the adhesive projectile slime of velvet worms

天鹅绒虫粘性喷射黏液中保守的富含亮氨酸重复序列蛋白

Hu, Zhaolong; Baer, Alexander; Hering, Lars; de Sena Oliveira, Ivo; Poulhazan, Alexandre; Browne, Darren C; Guo, Xue; Perrin, Quentin Moana; Sobota, Radoslaw M; Hoon, Shawn; Mayer, Georg; Kannan, Srinivasaraghavan; Verma, Chandra S; Harrington, Matthew J; Miserez, Ali

Responsiveness of different MET tumour alterations to type I and type II MET inhibitors.

不同MET肿瘤改变对I型和II型MET抑制剂的反应性

Murciano-Goroff Yonina R, Foglizzo Valentina, Chang Jason, Rekhtman Natasha, Sisk Ann Elizabeth, Gibson Jamie, Judka Lia, Clemens Kristen, Roa Paola, Ahmed Shaza Sayed, Bremer Nicole V, Binaco Courtney Lynn, Muzungu Sherifah Kemigisha, Rodriguez Estelamari, Merrill Madeline, Sgroe Erica, Repetto Matteo, Stadler Zsofia K, Berger Michael F, Yu Helena A, Toska Eneda, Kannan Srinivasaraghavan, Verma Chandra S, Drilon Alexander, Cocco Emiliano

Expanding the DNA editing toolbox: Novel lambda integrase variants targeting microalgal and human genome sequences

拓展DNA编辑工具箱:靶向微藻和人类基因组序列的新型λ整合酶变体

Siau, Jia Wei; Siddiqui, Asim Azhar; Lau, Sze Yi; Kannan, Srinivasaraghavan; Peter, Sabrina; Zeng, Yingying; Verma, Chandra; Droge, Peter; Ghadessy, John F

Rarγ -Foxa1 signaling promotes luminal identity in prostate progenitors and is disrupted in prostate cancer

Rarγ-Foxa1信号通路促进前列腺祖细胞的管腔特性,并在前列腺癌中受到破坏。

Felice, Dario De; Alaimo, Alessandro; Bressan, Davide; Genovesi, Sacha; Marmocchi, Elisa; Annesi, Nicole; Beccaceci, Giulia; Dalfovo, Davide; Cutrupi, Federico; Foletto, Veronica; Lorenzoni, Marco; Gandolfi, Francesco; Kannan, Srinivasaraghavan; Verma, Chandra S; Vasciaveo, Alessandro; Shen, Michael M; Romanel, Alessandro; Chiacchiera, Fulvio; Cambuli, Francesco; Lunardi, Andrea

Stitched peptides as potential cell permeable inhibitors of oncogenic DAXX protein.

拼接肽作为致癌DAXX蛋白的潜在细胞渗透性抑制剂

Jelinska Clare, Kannan Srinivasaraghavan, Frosi Yuri, Ramlan Siti Radhiah, Winnerdy Fernaldo, Lakshminarayanan Rajamani, Johannes Charles W, Brown Christopher J, Phan Anh-Tuan, Rhodes Daniela, Verma Chandra S

Author Correction: High p16 expression and heterozygous RB1 loss are biomarkers for CDK4/6 inhibitor resistance in ER(+) breast cancer

作者更正:p16高表达和RB1杂合缺失是ER(+)乳腺癌中CDK4/6抑制剂耐药的生物标志物。

Palafox, Marta; Monserrat, Laia; Bellet, Meritxell; Villacampa, Guillermo; Gonzalez-Perez, Abel; Oliveira, Mafalda; Brasó-Maristany, Fara; Ibrahimi, Nusaibah; Kannan, Srinivasaraghavan; Mina, Leonardo; Herrera-Abreu, Maria Teresa; Òdena, Andreu; Sánchez-Guixé, Mònica; Capelán, Marta; Azaro, Analía; Bruna, Alejandra; Rodríguez, Olga; Guzmán, Marta; Grueso, Judit; Viaplana, Cristina; Hernández, Javier; Su, Faye; Lin, Kui; Clarke, Robert B; Caldas, Carlos; Arribas, Joaquín; Michiels, Stefan; García-Sanz, Alicia; Turner, Nicholas C; Prat, Aleix; Nuciforo, Paolo; Dienstmann, Rodrigo; Verma, Chandra S; Lopez-Bigas, Nuria; Scaltriti, Maurizio; Arnedos, Monica; Saura, Cristina; Serra, Violeta

Activation of p53: How phosphorylated Ser15 triggers sequential phosphorylation of p53 at Thr18 by CK1δ

p53 的激活:磷酸化的 Ser15 如何触发 CK1δ 对 p53 在 Thr18 位点的连续磷酸化

Nicolaou, Sonia T; Kannan, Srinivasaraghavan; Warwicker, Jim; Verma, Chandra S

Discovery of cell active macrocyclic peptides with on-target inhibition of KRAS signaling

发现具有靶向抑制KRAS信号通路活性的细胞活性大环肽

Lim, Shuhui; Boyer, Nicolas; Boo, Nicole; Huang, Chunhui; Venkatachalam, Gireedhar; Angela Juang, Yu-Chi; Garrigou, Michael; Kaan, Hung Yi Kristal; Duggal, Ruchia; Peh, Khong Ming; Sadruddin, Ahmad; Gopal, Pooja; Yuen, Tsz Ying; Ng, Simon; Kannan, Srinivasaraghavan; Brown, Christopher J; Verma, Chandra S; Orth, Peter; Peier, Andrea; Ge, Lan; Yu, Xiang; Bhatt, Bhavana; Chen, Feifei; Wang, Erjia; Li, Nianyu Jason; Gonzales, Raymond J; Stoeck, Alexander; Henry, Brian; Sawyer, Tomi K; Lane, David P; Johannes, Charles W; Biswas, Kaustav; Partridge, Anthony W